SCHEMBL27897828

SCHEMBL27897828

O=CC1Cc2cc([N+](=O)[O-])ccc2N1

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PNMT P11086 10/20 0.45
ADRA2A P08913 7/20 0.45
ADRA2B P18089 3/20 0.45
ADRA2C P18825 3/20 0.45
ALDH1A1 P00352 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27799204 0.85 SIRT2 (0.45) PNMTADRA2AADRA2BADRA2CALDH1A1
SCHEMBL28431711 0.83 SIRT2 (0.43) PNMTADRA2AADRA2BADRA2CALDH1A1
SCHEMBL13362059 0.82 PNMT (0.52) PNMTADRA2AADRA2BADRA2CALDH1A1
SCHEMBL257552 0.78 ALDH1A1 (0.62) PNMTADRA2AADRA2BADRA2CALDH1A1
SCHEMBL6968655 0.78 ALDH1A1 (0.62) PNMTADRA2AADRA2BADRA2CALDH1A1
SCHEMBL28239780 0.78 PNMT (0.47) PNMTADRA2AADRA2BADRA2CALDH1A1
SCHEMBL27602097 0.77 SNCA (0.43) ALDH1A1SMN1; SMN2
SCHEMBL13222799 0.76 PNMT (0.40) PNMTADRA2AADRA2BADRA2CALDH1A1
SCHEMBL13062867 0.76 PNMT (0.44) PNMTADRA2AADRA2BADRA2CALDH1A1
SCHEMBL27587569 0.75 CHRNB4 (0.39) ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108822017-A New indole ketone compound and its preparation method and medicinal usage 中国医学科学院药物研究所 2018-11-16 CN claimed
CN-102797043-B Medicinal molecular fragment library and construction process thereof Tianli (Tianjin) Technology Co., Ltd. (CN) 2015-11-25 CN claimed
CN-104774193-A Indolone compounds as well as preparation method and medical application thereof UNIV CHINA PHARMA 2015-07-15 CN claimed
CN-102797043-A Medicinal molecular fragment library and construction method thereof CBB NETWORK CO LTD 2012-11-28 CN claimed
CN-108822017-A New indole ketone compound and its preparation method and medicinal usage 中国医学科学院药物研究所 2018-11-16 CN disclosed
CN-102797043-B Medicinal molecular fragment library and construction process thereof Tianli (Tianjin) Technology Co., Ltd. (CN) 2015-11-25 CN disclosed
CN-104774193-A Indolone compounds as well as preparation method and medical application thereof UNIV CHINA PHARMA 2015-07-15 CN disclosed
CN-102797043-A Medicinal molecular fragment library and construction method thereof CBB NETWORK CO LTD 2012-11-28 CN disclosed