SCHEMBL27900484

SCHEMBL27900484

CCCC[S+]([O-])NCc1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.42
POLB P06746 1/20 0.42
KDM4E B2RXH2 1/20 0.41
CYP3A4 P08684 1/20 0.41
MAPT P10636 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.39
ALPL P05186 1/20 0.39
GAA P10253 1/20 0.39
HPGD P15428 1/20 0.39
ALOX12 P18054 1/20 0.39
MAOA P21397 1/20 0.38
IDO1 P14902 2/20 0.38
THRB P10828 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
CNR2 P34972 1/20 0.37
CHRM2 P08172 1/20 0.37
CASP6 P55212 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28665142 0.78 IDO1 (0.44) POLBKDM4ECYP3A4MAPTGAA
SCHEMBL18602719 0.78 CYP3A4 (0.48) KDM4ECYP3A4MAPTSIGMAR1HPGD
SCHEMBL11064796 0.77 TDP1 (0.41) POLBKDM4ECYP3A4MAPTGAA
SCHEMBL11061936 0.77 IDO1 (0.40) POLBKDM4ECYP3A4MAPTGAA
SCHEMBL13616530 0.76 CES2 (0.38) MAPTSIGMAR1GAAMEN1KMT2A
SCHEMBL19785138 0.74 MEN1 (0.42) KDM4ECYP3A4MAPTSIGMAR1GAA
SCHEMBL17104769 0.73 TP53 (0.39) EPHX2SIGMAR1SMN1; SMN2MEN1KMT2A
SCHEMBL779932 0.72 CES2 (0.37) SIGMAR1SMN1; SMN2TDP1TP53TSHR
SCHEMBL9760714 0.72 CES2 (0.37) SIGMAR1SMN1; SMN2TDP1TP53TSHR
SCHEMBL30828004 0.72 CES2 (0.37) SIGMAR1SMN1; SMN2TDP1TP53TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103030656-B The synthetic method of proteasome inhibitor bortezomib and analogue thereof PEKING UNIVERSITY (CN) 2015-08-26 CN disclosed
CN-103030656-A Synthetic method of proteasome inhibitor bortezomib and analogs UNIV BEIJING 2013-04-10 CN disclosed