SCHEMBL27900613

SCHEMBL27900613

Cc1cccc(C(=O)c2cccc(C)c2-n2nccn2)c1-n1nccn1

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 17/20 0.50
HCRTR2 O43614 16/20 0.50
CYP3A4 P08684 6/20 0.43
ELANE P08246 1/20 0.42
CYP2C9 P11712 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17071985 0.88 HCRTR1 (0.49) HCRTR1HCRTR2CYP3A4ELANE
SCHEMBL31175258 0.88 KDM4E (0.50) HCRTR1HCRTR2CYP3A4CYP2C9KMT2A
SCHEMBL1586785 0.88 KDM4E (0.50) HCRTR1HCRTR2CYP3A4CYP2C9KMT2A
SCHEMBL17069778 0.83 HCRTR1 (0.46) HCRTR1HCRTR2CYP3A4
SCHEMBL14886143 0.80 ALDH1A1 (0.41) HCRTR1HCRTR2CYP3A4KMT2A
SCHEMBL27883288 0.79 HCRTR1 (0.48) HCRTR1HCRTR2
SCHEMBL27883266 0.73 HCRTR1 (0.54) HCRTR1HCRTR2CYP3A4ELANECYP2C9
SCHEMBL14951333 0.72 P2RX7 (0.36) HCRTR1HCRTR2CYP3A4KMT2A
SCHEMBL14886142 0.72 ACHE (0.43) HCRTR1HCRTR2CYP3A4KMT2A
SCHEMBL24013355 0.71 HCRTR1 (0.36) HCRTR1HCRTR2CYP3A4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102781942-A Disubstituted octahy-dropyrrolo [3,4-c]pyrroles as orexin receptor modulators JANSSEN PHARMACEUTICA NV 2012-11-14 CN claimed
CN-102781942-A Disubstituted octahy-dropyrrolo [3,4-c]pyrroles as orexin receptor modulators JANSSEN PHARMACEUTICA NV 2012-11-14 CN disclosed