SCHEMBL27900652

SCHEMBL27900652

CC(C)Nc1nccc(CC(C(=O)C(Cc2ccnc(NC(C)C)n2)c2ccc(F)cc2)c2ccc(F)cc2)n1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 3/20 0.41
ADRA1D P25100 2/20 0.41
ADRA1A P35348 2/20 0.41
ADRA1B P35368 2/20 0.41
HTR2C P28335 1/20 0.41
IDH1 O75874 5/20 0.39
NTRK1 P04629 1/20 0.39
KCNH3 Q9ULD8 1/20 0.39
ACACB O00763 1/20 0.39
PDE6D O43924 2/20 0.38
KRAS P01116 1/20 0.38
MAPK14 Q16539 6/20 0.38
MAPK13 O15264 3/20 0.38
MAPK12 P53778 3/20 0.38
MAPK11 Q15759 3/20 0.38
MAPK1 P28482 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1554350 0.79 RAB9A (0.50) HTR7ADRA1DADRA1AADRA1BHTR2C
SCHEMBL27883340 0.78 GRM5 (0.38)
SCHEMBL27522099 0.77 ALDH1A1 (0.43) ACACBMAPK14MAPK13MAPK12MAPK11
SCHEMBL22387976 0.75 HRH4 (0.45) HTR7IDH1KCNH3ACACBMAPK1
SCHEMBL15357780 0.73 HRH4 (0.46) HTR7KCNH3ACACBMAPK14
SCHEMBL12411105 0.72 HRH4 (0.45) HTR7IDH1KCNH3ACACBMAPK14
SCHEMBL28757676 0.72 KCNH3 (0.42) KCNH3MAPK14
SCHEMBL22388247 0.70 HRH4 (0.44) HTR7ACACB
SCHEMBL709768 0.70 CES1 (0.43) IDH1KCNH3MAPK14MAPK1
SCHEMBL27989070 0.69 KDM4E (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102834387-A Phenylpyri(mi)dinylpyrazoles and their use as fungicides BAYER CROPSCIENCE AG 2012-12-19 CN disclosed