SCHEMBL27901796

SCHEMBL27901796

O=CC1NCCc2ccc(C(F)(F)F)cc21

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.54
HTR2C P28335 3/20 0.54
HTR2B P41595 3/20 0.54
PARP1 P09874 1/20 0.46
PARP10 Q53GL7 1/20 0.46
KDM1A O60341 4/20 0.44
PNMT P11086 4/20 0.39
CHRNB2 P17787 2/20 0.39
CHRNA4 P43681 2/20 0.39
CHRNB4 P30926 1/20 0.39
CHRNA3 P32297 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.37
TDP2 O95551 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27901789 0.88 KDM1A (0.47) HTR2AHTR2CHTR2BPARP1PARP10
SCHEMBL27919503 0.80 OPRM1 (0.43) HTR2AHTR2CHTR2BKDM1A
SCHEMBL27919507 0.77 HTR2C (0.50) HTR2AHTR2CHTR2BPARP1PARP10
SCHEMBL27797441 0.77 HTR2A (0.50) HTR2AHTR2CHTR2BPARP1PARP10
SCHEMBL27743677 0.77 DRD2 (0.44) KDM1A
SCHEMBL27919637 0.77 TBXA2R (0.37) HTR2AHTR2CHTR2BCHRNB2CHRNA4
SCHEMBL1011414 0.77 HTR2A (0.66) HTR2AHTR2CHTR2BPARP1PARP10
SCHEMBL27901793 0.75 PRCP (0.42) HTR2AHTR2CHTR2BPARP1PARP10
SCHEMBL27901797 0.74 HTR2C (0.45) HTR2AHTR2CHTR2BPARP1PARP10
SCHEMBL27919511 0.74 HTR2C (0.36) HTR2AHTR2CHTR2BKDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103108871-B 17a-hydroxylase/c17,20-lyase inhibitors NOVARTIS AG 2014-09-10 CN disclosed
CN-103108871-A 17a-hydroxylase/c17,20-lyase inhibitors NOVARTIS AG 2013-05-15 CN disclosed