SCHEMBL27797441

SCHEMBL27797441

O=CC1NCCc2ccc(Br)cc21

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.50
HTR2C P28335 4/20 0.50
HTR2B P41595 3/20 0.50
PARP10 Q53GL7 2/20 0.41
PARP1 P09874 1/20 0.41
PNMT P11086 2/20 0.41
ASIC3 Q9UHC3 1/20 0.41
KDM1A O60341 4/20 0.40
PARP11 Q9NR21 1/20 0.38
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27708455 0.87 KDM1A (0.43) HTR2AHTR2CHTR2BPARP10PARP1
SCHEMBL27780964 0.83 PNMT (0.44) HTR2AHTR2CHTR2BPNMTASIC3
SCHEMBL27919637 0.81 TBXA2R (0.37) HTR2AHTR2CHTR2B
SCHEMBL27743677 0.81 DRD2 (0.44) KDM1A
SCHEMBL27919507 0.81 HTR2C (0.50) HTR2AHTR2CHTR2BPARP10PARP1
SCHEMBL28823708 0.78 CAMK2A (0.47) HTR2AHTR2CHTR2BPARP10PARP1
SCHEMBL27901796 0.77 HTR2A (0.54) HTR2AHTR2CHTR2BPARP10PARP1
SCHEMBL27779522 0.77 F2 (0.38) HTR2AHTR2CHTR2B
SCHEMBL95059 0.76 PRCP (0.53) HTR2AHTR2CHTR2B
SCHEMBL1799182 0.76 PRCP (0.53) HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113811529-A Fibroblast activation protein inhibitor 普拉西斯生物技术有限责任公司 2021-12-17 CN disclosed
CN-103108871-B 17a-hydroxylase/c17,20-lyase inhibitors NOVARTIS AG 2014-09-10 CN disclosed
CN-103108871-A 17a-hydroxylase/c17,20-lyase inhibitors NOVARTIS AG 2013-05-15 CN disclosed
CN-101848896-A Isoquinolinyl and isoindolinyl derivatives as histamine-3 antagonists WYETH CORP 2010-09-29 CN disclosed