SCHEMBL27901952

SCHEMBL27901952

O=CC1c2ccc(F)cc2CCN1c1cnccc1C(F)(F)F

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 5/20 0.37
TRPM8 Q7Z2W7 2/20 0.36
TRPA1 O75762 1/20 0.35
CYP17A1 P05093 6/20 0.33
SCD O00767 1/20 0.33
RBP4 P02753 1/20 0.33
C5AR1 P21730 1/20 0.33
CYP19A1 P11511 2/20 0.32
CYP11B1 P15538 2/20 0.32
TRPV1 Q8NER1 1/20 0.32
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27919502 0.88 CYP11B2 (0.36) CYP11B2CYP17A1RBP4C5AR1HTR2A
SCHEMBL27901787 0.84 CYP11B2 (0.35) CYP11B2CYP17A1SCDCYP11B1
SCHEMBL27919520 0.84 HTR2C (0.43) CYP11B2CYP17A1RBP4HTR2AHTR2C
SCHEMBL27919506 0.83 CYP17A1 (0.45) CYP17A1
SCHEMBL27901758 0.83 HTR2A (0.39) CYP11B2TRPM8CYP17A1SCDHTR2A
SCHEMBL27919510 0.81 CYP11B2 (0.35) CYP11B2CYP17A1C5AR1HTR2AHTR2C
SCHEMBL27919589 0.81 CYP11B2 (0.33) CYP11B2TRPM8C5AR1
SCHEMBL27919566 0.80 CYP11B2 (0.33) CYP11B2TRPM8RBP4C5AR1HTR2A
SCHEMBL27919635 0.78 SIRT6 (0.36) CYP11B2C5AR1HTR2AHTR2C
SCHEMBL27901761 0.77 HTR2C (0.39) CYP11B2TRPM8CYP17A1SCDCYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103108871-A 17a-hydroxylase/c17,20-lyase inhibitors NOVARTIS AG 2013-05-15 CN disclosed