SCHEMBL27905445

SCHEMBL27905445

CC(=O)Oc1nc(Br)ccc1N

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.36
LMNA P02545 1/20 0.33
MAPT P10636 5/20 0.32
POLB P06746 4/20 0.32
GLA P06280 3/20 0.32
KDM4E B2RXH2 2/20 0.32
CA12 O43570 1/20 0.32
GAA P10253 1/20 0.32
CA9 Q16790 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
CYP19A1 P11511 1/20 0.32
NPC1 O15118 1/20 0.32
MAPK1 P28482 1/20 0.32
HTT P42858 1/20 0.32
CFD P00746 1/20 0.32
FLT3 P36888 1/20 0.31
ADORA2A P29274 1/20 0.31
PKM P14618 1/20 0.31
ALDH1A1 P00352 1/20 0.30
F2 P00734 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2722243 0.84 KDM4E (0.35) MAPTPOLBGLAKDM4E
SCHEMBL2723798 0.83 HSD17B10 (0.33) MAPTPOLBGLAKDM4EGAA
SCHEMBL27850349 0.80 GRM5 (0.40) ALOX5LMNAMAPTPOLBGLA
SCHEMBL28783444 0.79 ALOX5 (0.36) ALOX5LMNAMAPTPOLBGLA
SCHEMBL27543527 0.79 KDM4E (0.39) ALOX5LMNAMAPTKDM4ETDP1
SCHEMBL27517890 0.75 ATR (0.39) ALOX5GLACYP19A1HTTALDH1A1
SCHEMBL156162 0.75 IDO1 (0.36) MAPTPOLBTDP1NPC1ALDH1A1
SCHEMBL29948393 0.75 IDO1 (0.36) MAPTPOLBTDP1NPC1ALDH1A1
SCHEMBL27543750 0.75 NQO2 (0.33) ALOX5MAPK1
SCHEMBL17753601 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103153997-B Quinazoline derivatives MERCK PATENT GMBH 2015-04-29 CN disclosed
CN-103429572-A Tetra-substituted cyclohexyl compounds as kinase inhibitors NOVARTIS AG 2013-12-04 CN disclosed
CN-103153997-A Quinazoline derivatives MERCK PATENT GMBH 2013-06-12 CN disclosed
CN-103080106-A Cyclic ether compounds useful as kinase inhibitors NOVARTIS AG 2013-05-01 CN disclosed