SCHEMBL27912640

SCHEMBL27912640

COC(=O)c1nn(CC(F)(F)F)cc1N

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CFTR P13569 3/20 0.36
ADORA3 P0DMS8 2/20 0.36
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
NPSR1 Q6W5P4 1/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
CYP1A2 P05177 1/20 0.35
KDM4E B2RXH2 4/20 0.34
HTT P42858 2/20 0.34
TP53 P04637 1/20 0.34
POLB P06746 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
ALDH1A1 P00352 2/20 0.33
MAP3K5 Q99683 1/20 0.33
NPC1 O15118 1/20 0.33
KMT2A Q03164 1/20 0.33
RAB9A P51151 1/20 0.33
PDE10A Q9Y233 1/20 0.33
HDAC9 Q9UKV0 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28946943 0.86 CFTR (0.35) CFTRNPSR1SMN1; SMN2CYP1A2KDM4E
SCHEMBL31429362 0.82 NPC1 (0.46) SMN1; SMN2KDM4EHTTALDH1A1NPC1
SCHEMBL7510800 0.82 PDE10A (0.42) CFTRADORA3ADORA2AADORA1SMN1; SMN2
SCHEMBL3059091 0.81 ALDH1A1 (0.50) NPSR1SMN1; SMN2CYP1A2KDM4EHTT
SCHEMBL7509900 0.79 PDE10A (0.41) ADORA3ADORA2AADORA1SMN1; SMN2KDM4E
SCHEMBL27912638 0.79 ALDH1A1 (0.45) SMN1; SMN2KDM4EHTTPOLBALDH1A1
SCHEMBL1664763 0.78 LRRK2 (0.37) MAP3K5PDE10A
SCHEMBL19208770 0.76 ENPP2 (0.36) ADORA3ADORA2AADORA1NPSR1SMN1; SMN2
SCHEMBL17459117 0.75 KMT2A (0.43) NPSR1SMN1; SMN2CYP1A2KDM4EHTT
Dimethylformamide SCHEMBL27895442 0.75 ADORA3 (0.32) ADORA3PDE10AHDAC9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102947292-A nitrogen-containing heteroaryl compounds HOFFMANN LA ROCHE 2013-02-27 CN disclosed