SCHEMBL27919782

SCHEMBL27919782

COc1ccccc1C(C#N)Cc1cc(C)cc(C)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.40
ESR1 P03372 1/20 0.40
ESR2 Q92731 1/20 0.40
SGMS2 Q8NHU3 5/20 0.40
KDM4E B2RXH2 2/20 0.40
CYP2C19 P33261 3/20 0.37
LMNA P02545 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
L3MBTL1 Q9Y468 2/20 0.36
POLB P06746 1/20 0.36
HTT P42858 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
CTSB P07858 2/20 0.36
GAA P10253 1/20 0.36
CTSL P07711 1/20 0.36
CTSS P25774 1/20 0.36
IDH1 O75874 1/20 0.35
CYP2D6 P10635 1/20 0.35
MAPT P10636 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27916171 0.84 SGMS2 (0.49) ALDH1A1ESR1ESR2SGMS2KDM4E
SCHEMBL9229299 0.80 TAAR1 (0.51) ALDH1A1SGMS2KDM4ECYP2C19LMNA
SCHEMBL27919783 0.73 TACR1 (0.39) CYP2C19L3MBTL1POLBHTTNPSR1
SCHEMBL9450168 0.72 SYK (0.43) ALDH1A1SGMS2KDM4EL3MBTL1
SCHEMBL30366298 0.72 ESR2 (0.43) ALDH1A1ESR1ESR2CYP2C19LMNA
SCHEMBL28618652 0.70 ESR2 (0.46) ALDH1A1ESR1ESR2CYP2C19CYP1A2
SCHEMBL18284609 0.70 PPARG (0.40) ALDH1A1SGMS2KDM4EL3MBTL1POLB
SCHEMBL21632015 0.70 L3MBTL1 (0.55) ALDH1A1SGMS2KDM4ELMNAL3MBTL1
SCHEMBL10399399 0.70 TP53 (0.40) ALDH1A1KDM4ECYP2C19LMNAL3MBTL1
SCHEMBL21632162 0.69 POLB (0.50) ALDH1A1SGMS2KDM4ELMNAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103339095-A Alkyne and alkene derivatives as sphingosine 1-phosphate-1 receptor modulators ALLERGAN INC 2013-10-02 CN disclosed