SCHEMBL9229299

SCHEMBL9229299

COc1cccc(CC(C#N)c2ccccc2OC)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.51
ABCB1 P08183 6/20 0.44
KMT2A Q03164 2/20 0.43
HTR1A P08908 3/20 0.43
DRD2 P14416 2/20 0.43
MEN1 O00255 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
RECQL P46063 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
IDO1 P14902 2/20 0.42
AGXT P21549 2/20 0.42
ALDH1A1 P00352 2/20 0.42
SGMS2 Q8NHU3 2/20 0.42
LMNA P02545 1/20 0.42
GAA P10253 1/20 0.42
MAOB P27338 1/20 0.41
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27916171 0.85 SGMS2 (0.49) CYP1A2CYP2C9CYP2C19L3MBTL1IDO1
SCHEMBL27919782 0.80 ALDH1A1 (0.40) CYP1A2CYP2C9CYP2C19L3MBTL1ALDH1A1
SCHEMBL1442239 0.77 TAAR1 (0.62) TAAR1IDO1AGXTMAOB
SCHEMBL620934 0.77 CASR (0.52) TAAR1KMT2ASGMS2MAOB
SCHEMBL9230601 0.75 TAAR1 (0.51) TAAR1ABCB1KMT2AHTR1ADRD2
SCHEMBL9228226 0.75 TAAR1 (0.51) TAAR1ABCB1KMT2AHTR1ADRD2
SCHEMBL8417617 0.75 TAAR1 (0.58) TAAR1CYP1A2IDO1AGXT
SCHEMBL623518 0.74 KMT2A (0.43) TAAR1KMT2AHTR1AL3MBTL1ALDH1A1
SCHEMBL9230011 0.74 TAAR1 (0.54) TAAR1ABCB1KMT2AHTR1ADRD2
SCHEMBL7872355 0.74 ABCB1 (0.54) ABCB1HTR1ADRD2ALDH1A1SGMS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661266-A1 Substituted cyclic amine compounds as 5HT2 antagonists TOA EIYO LTD. (JP) 1995-07-05 EP disclosed