SCHEMBL27922016

SCHEMBL27922016

CC(=O)C=C(c1ccccc1)c1ccccc1.[Pd].[Pd]

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.48
MTNR1B P49286 1/20 0.48
CES2 O00748 3/20 0.48
CES1 P23141 3/20 0.48
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
NFE2L2 Q16236 1/20 0.45
ALDH1A1 P00352 4/20 0.44
TSHR P16473 3/20 0.44
DAO P14920 1/20 0.44
NAPRT Q6XQN6 1/20 0.44
TDP1 Q9NUW8 3/20 0.43
CA12 O43570 2/20 0.43
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA9 Q16790 2/20 0.43
GLA P06280 1/20 0.43
MAPK1 P28482 1/20 0.43
AKT1 P31749 1/20 0.41
MAPT P10636 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27589809 1.00 MTNR1A (0.48) MTNR1AMTNR1BCES2CES1MEN1
SCHEMBL28385832 1.00 MTNR1A (0.48) MTNR1AMTNR1BCES2CES1MEN1
SCHEMBL27498418 1.00 MTNR1A (0.48) MTNR1AMTNR1BCES2CES1MEN1
SCHEMBL4863098 0.98 CES2 (0.50) MTNR1AMTNR1BCES2CES1MEN1
SCHEMBL27573431 0.95 MTNR1A (0.48) MTNR1AMTNR1BCES2CES1MEN1
Chloroform SCHEMBL5461181 0.94 MTNR1A (0.44) MTNR1AMTNR1BCES2CES1MEN1
SCHEMBL27962243 0.86 TDP1 (0.44) MTNR1AMTNR1BCES2CES1MEN1
SCHEMBL25252302 0.82 NR4A1 (0.58) CES2CES1ALDH1A1TSHRCYP2C19
Tromethamine SCHEMBL21616749 0.82 MTNR1A (0.42) MTNR1AMTNR1BCES2CES1MEN1
Tromethamine SCHEMBL5461179 0.80 MTNR1A (0.39) MTNR1AMTNR1BCES2CES1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115052873-A Heteroaromatic carboxamide derivatives as plasma kallikrein inhibitors 勃林格殷格翰国际有限公司 2022-09-13 CN disclosed
CN-111362975-B Naphthyridine compounds as JAK kinase inhibitors 施万生物制药研发IP有限责任公司 2022-04-05 CN disclosed
CN-103502228-A Novel photoactive polymers MERCK PATENT GMBH 2014-01-08 CN disclosed
CN-103140479-A Process for producing pyrimidine derivative NOVARTIS AG 2013-06-05 CN disclosed