SCHEMBL27934811

SCHEMBL27934811

O=C(NCc1cccs1)c1ncccc1O

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.68
EGLN2 Q96KS0 1/20 0.57
FTO Q9C0B1 1/20 0.57
HPGD P15428 7/20 0.56
ALDH1A1 P00352 4/20 0.52
TSHR P16473 2/20 0.52
HSD17B10 Q99714 1/20 0.52
POLB P06746 1/20 0.51
KMT2A Q03164 3/20 0.51
MEN1 O00255 2/20 0.51
LMNA P02545 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
MAPT P10636 2/20 0.50
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
HTT P42858 1/20 0.50
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16598147 0.77 HPGD (0.61) KDM4EHPGDALDH1A1TSHRHSD17B10
SCHEMBL1722407 0.77 KDM4E (0.70) KDM4EHPGDALDH1A1TSHRHSD17B10
SCHEMBL12907922 0.77 KDM4E (0.70) KDM4EHPGDALDH1A1TSHRHSD17B10
SCHEMBL27815171 0.77 KDM4E (0.70) KDM4EHPGDALDH1A1TSHRHSD17B10
SCHEMBL31026221 0.77 EGLN2 (0.68) EGLN2FTOALDH1A1KMT2AHTT
SCHEMBL15327067 0.76 KDM4E (0.59) KDM4EHPGDALDH1A1TSHRHSD17B10
SCHEMBL2201945 0.76 EGLN1 (0.66) KDM4EHPGDALDH1A1HSD17B10POLB
SCHEMBL27949742 0.75 ALDH1A1 (0.62) KDM4EEGLN2FTOHPGDALDH1A1
SCHEMBL30927143 0.75 ALDH1A1 (0.62) KDM4EEGLN2FTOHPGDALDH1A1
SCHEMBL24405087 0.75 FTO (0.65) KDM4EEGLN2FTOALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103539731-B Amides compound of pyridine 2 and preparation method thereof, its pharmaceutical composition and purposes 中国科学院上海药物研究所 2018-01-05 CN disclosed
CN-103539731-A Pyridine-2-amide compound as well as preparation method, pharmaceutical composition and use thereof SHANGHAI INST MATERIA MEDICA 2014-01-29 CN disclosed