SCHEMBL27944239

SCHEMBL27944239

NC(=O)c1[nH]ccc1-c1cc(F)cc(F)c1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.39
MAP2 P11137 2/20 0.36
SLC9A1 P19634 2/20 0.35
HPGDS O60760 1/20 0.35
IKBKB O14920 2/20 0.35
PARP1 P09874 1/20 0.34
CCNC P24863 4/20 0.34
CDK8 P49336 4/20 0.34
CDC7 O00311 3/20 0.33
PIK3CD O00329 1/20 0.33
PIK3CA P42336 1/20 0.33
PIK3CB P42338 1/20 0.33
CHUK O15111 1/20 0.33
CES2 O00748 1/20 0.32
CES1 P23141 1/20 0.32
PRKCI P41743 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28202946 0.85 HPGDS (0.48) MAP2SLC9A1HPGDSPARP1CCNC
SCHEMBL27944229 0.79 MAP2 (0.41) MAP2SLC9A1IKBKBCCNCCDK8
SCHEMBL17604415 0.77 BCAT2 (0.50) BRD4MAP2IKBKBPARP1CCNC
SCHEMBL1925897 0.75 CCNC (0.39) IKBKBPARP1CCNCCDK8CHUK
SCHEMBL30471167 0.71
SCHEMBL1925356 0.69 TSHR (0.50) PARP1CDC7CES1
SCHEMBL3236362 0.68 BCAT2 (0.63) SLC9A1IKBKBPARP1CDC7
SCHEMBL17925960 0.68 BCL2L1 (0.47)
SCHEMBL562266 0.65
SCHEMBL6672416 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103649089-A Pyrrolotriazinones as PI3K inhibitors ALMIRALL SA 2014-03-19 CN disclosed