SCHEMBL27965451

SCHEMBL27965451

CCc1cc(NS(=O)(=O)CC2CN(C(c3ccc(Cl)cc3)c3ccc(Cl)cc3)C2)cc(C(=O)OF)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 3/20 0.36
SCN9A Q15858 3/20 0.34
CNR1 P21554 1/20 0.33
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
GPX4 P36969 2/20 0.32
SCN7A Q01118 1/20 0.31
SCN5A Q14524 1/20 0.31
KMT2A Q03164 1/20 0.31
CA12 O43570 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA9 Q16790 1/20 0.31
CACNA1G O43497 1/20 0.31
IDH1 O75874 1/20 0.31
ATM Q13315 1/20 0.31
MGLL Q99685 1/20 0.31
ABHD6 Q9BV23 1/20 0.31
NPC1 O15118 1/20 0.31
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL975275 0.84 SLC6A9 (0.39) SLC6A9CNR1OPRD1GPX4KMT2A
SCHEMBL975711 0.84 SLC6A9 (0.37) SLC6A9SCN9ACNR1OPRM1OPRD1
SCHEMBL977022 0.84 SLC6A9 (0.37) SLC6A9SCN9ACNR1OPRD1GPX4
SCHEMBL978430 0.83 HPGD (0.38) SLC6A9SCN9AOPRD1CA12CA1
SCHEMBL977237 0.82 SLC6A9 (0.37) SLC6A9OPRD1GPX4KMT2ACACNA1G
SCHEMBL976058 0.81 ATM (0.38) SLC6A9CNR1ATM
SCHEMBL979165 0.80 SLC6A9 (0.36) SLC6A9SCN9ACNR1OPRM1OPRD1
SCHEMBL975244 0.79 WDR5 (0.44) SLC6A9CNR1GPX4KMT2ACACNA1G
SCHEMBL974202 0.79 WDR5 (0.41) SLC6A9SCN9ACNR1GPX4SCN7A
SCHEMBL974408 0.79 WDR5 (0.41) SLC6A9SCN9ACNR1OPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101945852-B Azetidine derivatives, their preparation and their use in therapy SANOFI AVENTIS 2014-05-07 CN disclosed