SCHEMBL27969552

SCHEMBL27969552

Cc1cc(C)c(N(C)C(=O)OC(C)(C)C)c(C(=O)O)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.44
METAP2 P50579 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
CSNK2A1 P68400 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
BRD4 O60885 1/20 0.32
NFKB1 P19838 2/20 0.32
NFKB2 Q00653 2/20 0.32
RELA Q04206 2/20 0.32
STAT5B P51692 1/20 0.32
TPMT P51580 1/20 0.32
PAX8 Q06710 1/20 0.32
LCK P06239 1/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
ALDH1A1 P00352 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27969454 0.87 MYC (0.40) KDM4ECSNK2A1BRD4NFKB1NFKB2
SCHEMBL24072766 0.75 RXRB (0.42) NPSR1BRD4STAT5BPAX8MEN1
SCHEMBL30339105 0.75 RXRB (0.42) NPSR1BRD4STAT5BPAX8MEN1
SCHEMBL31716122 0.74 SSTR4 (0.37) KDM4EBRD4NFKB1NFKB2RELA
SCHEMBL31110212 0.72 ALDH1A1 (0.35) CYP2C19L3MBTL1STAT5BALDH1A1SMN1; SMN2
SCHEMBL22115129 0.72 ABL1 (0.38) CYP2C9CYP2C19NPSR1BRD4PAX8
SCHEMBL18091685 0.72 HSD17B10 (0.40) KDM4ENPSR1LCKMEN1KMT2A
SCHEMBL849774 0.72 CYP2C9 (0.34) KDM4ECYP2C9CYP2C19NPSR1BRD4
SCHEMBL27504065 0.70 KDM4E (0.50) KDM4EMETAP2CSNK2A1TPMTMEN1
SCHEMBL108498 0.70 LCK (0.50) KDM4EMETAP2L3MBTL1NFKB1NFKB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103992326-A Indol-hexahydropyrazine-quinazolinone anti-tumour compounds and preparation method thereof UNIV PLA 2ND MILITARY MEDICAL 2014-08-20 CN disclosed