SCHEMBL27969895

SCHEMBL27969895

Cn1cc(C(N)=O)c2c(CCC3CCCCC3)cccc21

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 6/20 0.44
SLC6A4 P31645 1/20 0.40
PARP2 Q9UGN5 3/20 0.40
CNR2 P34972 2/20 0.39
CNR1 P21554 2/20 0.39
RAB9A P51151 1/20 0.39
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
HTR2B P41595 1/20 0.38
CEL P19835 2/20 0.37
IL1B P01584 1/20 0.37
SIRT2 Q8IXJ6 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27969863 0.88 PARP1 (0.46) PARP1PARP2CNR2CNR1RAB9A
SCHEMBL27969898 0.87 PARP1 (0.44) PARP1PARP2CNR1RAB9AKMT2A
SCHEMBL27969862 0.86 CNR1 (0.43) PARP1PARP2CNR2CNR1KMT2A
SCHEMBL27969977 0.85 P2RX7 (0.48) PARP1PARP2CNR2CNR1KMT2A
SCHEMBL6175349 0.76 TP53 (0.43) RAB9AKMT2AMEN1CELSIRT2
SCHEMBL30100457 0.75 HMGB1 (0.44) PARP1RAB9AKMT2AMEN1CEL
SCHEMBL27969982 0.74 P2RX7 (0.53) PARP1CNR2CNR1KMT2AMEN1
SCHEMBL27969891 0.72 P2RX7 (0.51) PARP1CNR2CNR1KMT2AMEN1
SCHEMBL1020350 0.70 IL1B (0.53) CNR2CNR1RAB9AKMT2AIL1B
SCHEMBL1021986 0.70 IL1B (0.53) CNR2CNR1RAB9AKMT2AIL1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102046240-B Novel P2X7R antagonists and their use AFFECTIS PHARMACEUTICALS AG 2014-06-25 CN disclosed