SCHEMBL27972751

SCHEMBL27972751

CCC(C(=O)OC)c1ccc(N)c(F)c1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 11/20 0.43
AKR1C2 P52895 11/20 0.43
AKR1C1 Q04828 1/20 0.40
PTGS1 P23219 1/20 0.40
KCNQ2 O43526 1/20 0.40
ESR1 P03372 1/20 0.40
ESR2 Q92731 1/20 0.40
HDAC1 Q13547 3/20 0.40
HDAC6 Q9UBN7 1/20 0.40
SHBG P04278 1/20 0.38
HDAC3 O15379 2/20 0.37
HDAC2 Q92769 2/20 0.37
NCOR2 Q9Y618 2/20 0.37
DPP4 P27487 2/20 0.36
FOLH1 Q04609 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1590117 0.83 AKR1C3 (0.59) AKR1C3AKR1C2AKR1C1PTGS1
SCHEMBL24875589 0.82 AKR1C3 (0.43) AKR1C3AKR1C2AKR1C1PTGS1KCNQ2
SCHEMBL7708885 0.80 HDAC1 (0.42) HDAC1HDAC6DPP4FOLH1
SCHEMBL8476208 0.80 MT-CO2 (0.47) AKR1C3AKR1C2AKR1C1PTGS1HDAC1
SCHEMBL30192791 0.80 MT-CO2 (0.47) AKR1C3AKR1C2AKR1C1PTGS1HDAC1
SCHEMBL24875457 0.80 MT-CO2 (0.47) AKR1C3AKR1C2AKR1C1PTGS1HDAC1
SCHEMBL2295719 0.78 ESR1 (0.50) AKR1C3AKR1C2AKR1C1PTGS1ESR1
SCHEMBL13687168 0.78 ESR1 (0.50) KCNQ2ESR1ESR2
SCHEMBL3711505 0.78 HDAC1 (0.41) AKR1C3AKR1C2AKR1C1PTGS1HDAC1
SCHEMBL31478057 0.76 CPN1 (0.53) KCNQ2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103958472-A Aryl-or N-heteroaryl-substituted methanesulfonamide derivatives as vanilloid receptor ligands GRUENENTHAL GMBH 2014-07-30 CN disclosed