SCHEMBL27985191

SCHEMBL27985191

COC(=O)c1cccn2cccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.50
TSHR P16473 1/20 0.50
NR4A2 P43354 3/20 0.49
ALDH1A1 P00352 3/20 0.48
CFTR P13569 1/20 0.48
HSD17B10 Q99714 1/20 0.48
KDM4E B2RXH2 2/20 0.47
POLB P06746 1/20 0.47
ATM Q13315 1/20 0.47
KMT2A Q03164 6/20 0.46
MEN1 O00255 1/20 0.46
MYC P01106 1/20 0.46
MAPT P10636 3/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA5A P35218 1/20 0.43
CA9 Q16790 1/20 0.43
ALOX15 P16050 1/20 0.43
THRB P10828 1/20 0.43
GAA P10253 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3983002 0.89 NR4A2 (0.50) LMNATSHRNR4A2ALDH1A1CFTR
SCHEMBL25514681 0.80 PTGS2 (0.39) LMNATSHRNR4A2ALDH1A1CFTR
SCHEMBL25514677 0.75 ALDH1A1 (0.50) TSHRALDH1A1HSD17B10KDM4EPOLB
SCHEMBL8887417 0.75 LMNA (0.47) LMNATSHRNR4A2ALDH1A1CFTR
SCHEMBL20068336 0.75 MYC (0.49) LMNATSHRNR4A2ALDH1A1CFTR
SCHEMBL1878367 0.74 KDM4E (0.49) LMNATSHRALDH1A1CFTRHSD17B10
Dimethyl Phthalate SCHEMBL29500970 0.74 TSHR (0.74) LMNATSHRALDH1A1CFTRHSD17B10
Dimethyl Phthalate SCHEMBL790124 0.74 TSHR (0.74) LMNATSHRALDH1A1CFTRHSD17B10
Dimethyl Phthalate SCHEMBL34630 0.74 TSHR (0.74) LMNATSHRALDH1A1CFTRHSD17B10
Dimethyl Phthalate SCHEMBL29669976 0.74 TSHR (0.74) LMNATSHRALDH1A1CFTRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117304130-A MCL-1 inhibitors 吉利德科学公司 2023-12-29 CN disclosed
CN-112118845-B MCL-1 inhibitors 吉利德科学公司 2023-06-13 CN disclosed
CN-110381738-B Pesticidal and parasiticidal vinyl isoxazoline compounds 勃林格殷格翰动物保健美国公司 2021-07-16 CN disclosed
CN-112118845-A MCL-1 inhibitors 吉利德科学公司 2020-12-22 CN disclosed
CN-104066330-A Isoxazoline derivatives for controlling ectoparasites LILLY CO ELI 2014-09-24 CN disclosed