SCHEMBL27985443

SCHEMBL27985443

Nc1nc(N)c(-c2cnccn2)c(-c2ccccn2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.46
ALOX15 P16050 2/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
ADORA2A P29274 4/20 0.44
ADORA1 P30542 3/20 0.44
ULK1 O75385 1/20 0.40
CDK7 P50613 1/20 0.40
CDK5 Q00535 1/20 0.40
PRKCE Q02156 1/20 0.40
CAMK2G Q13555 1/20 0.40
DYRK1A Q13627 1/20 0.40
CDK5R1 Q15078 1/20 0.40
RPS6KA1 Q15418 1/20 0.40
AAK1 Q2M2I8 1/20 0.40
MAP3K19 Q56UN5 1/20 0.40
CAMKK1 Q8N5S9 1/20 0.40
CAMKK2 Q96RR4 1/20 0.40
CYP2A6 P11509 1/20 0.39
F2 P00734 1/20 0.38
F12 P00748 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28791336 0.81 ADORA2A (0.48) ADORA2AADORA1CDK5CDK5R1CYP2A6
SCHEMBL27985752 0.81 ADORA2A (0.44) KDM4EADORA2AADORA1PRKCEDHFR
SCHEMBL27850416 0.81 HSP90AA1 (0.43) KDM4EALOX15L3MBTL1ADORA2AADORA1
SCHEMBL27985753 0.79 DHFR (0.33) KDM4EDHFRHTTMETAP2
Hydrochloric Acid SCHEMBL1367779 0.79 HSP90AA1 (0.41) KDM4EALOX15L3MBTL1ADORA2AADORA1
SCHEMBL27985373 0.75 DHFR (0.37) KDM4EADORA2AADORA1DHFRHSP90AA1
SCHEMBL28814482 0.74 ADORA2A (0.47) KDM4EADORA2AADORA1CYP2A6DHFR
SCHEMBL27985802 0.74 PIK3CD (0.35) KDM4EADORA2AADORA1DHFRHSP90AA1
SCHEMBL27831916 0.73 PIM1 (0.36) KDM4EADORA2ADHFRMAPK1
SCHEMBL5197687 0.73 KDM4E (0.44) KDM4EALOX15L3MBTL1ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102307869-B Aminopyrazine derivative and medicine NIPPON SHINYAKU CO.,LTD. (JP) 2014-10-22 CN claimed
CN-102307869-B Aminopyrazine derivative and medicine NIPPON SHINYAKU CO.,LTD. (JP) 2014-10-22 CN disclosed