SCHEMBL27985802

SCHEMBL27985802

Nc1nc(N)c(-c2cnccn2)c(-c2cncs2)n1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 2/20 0.35
PIK3CA P42336 2/20 0.35
PIK3CG P48736 2/20 0.35
PIK3CB P42338 1/20 0.35
PI4KA P42356 1/20 0.35
PI4KB Q9UBF8 1/20 0.35
ADORA2A P29274 3/20 0.33
ADORA1 P30542 3/20 0.33
HSP90AA1 P07900 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
ADORA2B P29275 1/20 0.33
KDM4E B2RXH2 1/20 0.32
GLA P06280 1/20 0.32
HTT P42858 1/20 0.31
RECQL P46063 1/20 0.31
DHFR P00374 1/20 0.31
PIM1 P11309 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27850416 0.78 HSP90AA1 (0.43) PIK3CDPIK3CAPIK3CGPIK3CBPI4KA
SCHEMBL28814482 0.78 ADORA2A (0.47) PIK3CDPIK3CAPIK3CGPIK3CBPI4KA
Hydrochloric Acid SCHEMBL1367779 0.77 HSP90AA1 (0.41) PIK3CDPIK3CAPIK3CGPIK3CBPI4KA
SCHEMBL27985752 0.75 ADORA2A (0.44) PIK3CDPIK3CAPIK3CGPIK3CBPI4KA
SCHEMBL27985443 0.74 KDM4E (0.46) ADORA2AADORA1HSP90AA1KDM4EHTT
SCHEMBL28791336 0.73 ADORA2A (0.48) ADORA2AADORA1HSP90AA1ADORA2BDHFR
SCHEMBL17201635 0.73 PIM1 (0.40) PIK3CDPIK3CAPIK3CGPIK3CBPI4KA
SCHEMBL27985753 0.71 DHFR (0.33) PIK3CDPIK3CAPIK3CGPIK3CBPI4KA
SCHEMBL27831916 0.71 PIM1 (0.36) PIK3CDPIK3CAPIK3CGPIK3CBPI4KA
SCHEMBL28814538 0.70 KDM4E (0.37) KDM4EGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102307869-B Aminopyrazine derivative and medicine NIPPON SHINYAKU CO.,LTD. (JP) 2014-10-22 CN claimed
CN-102307869-B Aminopyrazine derivative and medicine NIPPON SHINYAKU CO.,LTD. (JP) 2014-10-22 CN disclosed