SCHEMBL28814482

SCHEMBL28814482

Nc1nc(N)c(-c2cnccn2)c(-c2nccs2)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 8/20 0.47
ADORA1 P30542 8/20 0.47
HSP90AA1 P07900 1/20 0.41
CYP2A6 P11509 1/20 0.36
HTT P42858 1/20 0.34
RECQL P46063 1/20 0.34
ADORA3 P0DMS8 2/20 0.33
ADORA2B P29275 2/20 0.33
HDAC1 Q13547 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
PIK3CD O00329 1/20 0.32
PIK3CA P42336 1/20 0.32
PIK3CB P42338 1/20 0.32
PI4KA P42356 1/20 0.32
PIK3CG P48736 1/20 0.32
PI4KB Q9UBF8 1/20 0.32
DHFR P00374 3/20 0.32
KDM4E B2RXH2 1/20 0.32
GLA P06280 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27850416 0.78 HSP90AA1 (0.43) ADORA2AADORA1HSP90AA1HTTRECQL
SCHEMBL27985802 0.78 PIK3CD (0.35) ADORA2AADORA1HSP90AA1HTTRECQL
Hydrochloric Acid SCHEMBL1367779 0.77 HSP90AA1 (0.41) ADORA2AADORA1HSP90AA1HTTRECQL
SCHEMBL27985752 0.75 ADORA2A (0.44) ADORA2AADORA1HSP90AA1ADORA2BPIK3CD
SCHEMBL27985443 0.74 KDM4E (0.46) ADORA2AADORA1HSP90AA1CYP2A6HTT
SCHEMBL28791336 0.73 ADORA2A (0.48) ADORA2AADORA1HSP90AA1CYP2A6ADORA2B
SCHEMBL29791140 0.73 CYP2A6 (0.50) ADORA2AADORA1HSP90AA1CYP2A6HTT
SCHEMBL902694 0.73 CYP2A6 (0.50) ADORA2AADORA1HSP90AA1CYP2A6HTT
SCHEMBL1027238 0.71 CYP2A6 (0.48) ADORA2AADORA1HSP90AA1CYP2A6HTT
SCHEMBL27985753 0.71 DHFR (0.33) HTTRECQLPIK3CDPIK3CAPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102307869-B Aminopyrazine derivative and medicine NIPPON SHINYAKU CO.,LTD. (JP) 2014-10-22 CN claimed
CN-102307869-B Aminopyrazine derivative and medicine NIPPON SHINYAKU CO.,LTD. (JP) 2014-10-22 CN disclosed