SCHEMBL27987019

SCHEMBL27987019

CC[C@@H](CNc1nc(Cl)ncc1Cl)C(=N)C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
STK17B O94768 1/20 0.42
STK17A Q9UEE5 1/20 0.42
TDP1 Q9NUW8 1/20 0.32
TP53 P04637 2/20 0.31
MAPT P10636 2/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
THRB P10828 1/20 0.31
ALDH1A1 P00352 1/20 0.31
BCL6 P41182 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27987021 1.00 STK17B (0.42) STK17BSTK17ATDP1TP53MAPT
SCHEMBL28814671 0.78 STK17B (0.42) STK17BSTK17ABCL6
SCHEMBL27987449 0.78 ESR1 (0.33) ALDH1A1TSHR
SCHEMBL27987018 0.78 STK17B (0.42) STK17BSTK17ABCL6
SCHEMBL1937173 0.74 STK17A (0.41) STK17BSTK17AALDH1A1BCL6
SCHEMBL1937307 0.72 ESR1 (0.49) STK17BSTK17ATP53MAPTSMN1; SMN2
SCHEMBL27620523 0.71 RAB9A (0.38) TDP1SMN1; SMN2ALDH1A1
SCHEMBL5246243 0.70 STK17B (0.49) STK17BSTK17AMAPTALDH1A1
SCHEMBL1935303 0.70 STK17B (0.47) STK17BSTK17AALDH1A1
SCHEMBL20652230 0.69 STK17A (0.42) STK17BSTK17AALDH1A1BCL6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104169272-A Pyrimidine-2,4-diamine derivatives as kinase inhibitors CELLZOME LTD 2014-11-26 CN disclosed