SCHEMBL27993496

SCHEMBL27993496

CCSc1c(Cl)cccc1C#N

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.40
KDM4E B2RXH2 6/20 0.40
HPGD P15428 4/20 0.40
MAPT P10636 4/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
POLB P06746 2/20 0.40
STAT6 P42226 1/20 0.40
HIF1A Q16665 1/20 0.40
DYRK1A Q13627 1/20 0.38
TERT O14746 1/20 0.37
MAPK1 P28482 2/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 3/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
GAA P10253 1/20 0.35
LMNA P02545 2/20 0.35
PKM P14618 1/20 0.35
CLK1 P49759 1/20 0.35
S1PR1 P21453 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15389016 0.87 TSHR (0.41) ALDH1A1KDM4EHPGDMAPTMEN1
SCHEMBL7760077 0.80 TSHR (0.50) ALDH1A1KDM4EHPGDMAPTMEN1
SCHEMBL3780613 0.73 ALDH1A1 (0.38) ALDH1A1KDM4EHPGDMAPTMEN1
SCHEMBL16587420 0.72 DYRK1A (0.41) ALDH1A1KDM4EHPGDMAPTDYRK1A
SCHEMBL3790582 0.72 ALDH1A1 (0.47) ALDH1A1KDM4EHPGDMAPTMEN1
SCHEMBL4599675 0.69 AR (0.50) ALDH1A1KDM4EHPGDMAPTMEN1
SCHEMBL25483123 0.69 TAAR1 (0.39) ALDH1A1KDM4EHPGDMAPTDYRK1A
SCHEMBL102325 0.69 TSHR (0.48) ALDH1A1KDM4EHPGDDYRK1ATSHR
SCHEMBL30602897 0.68 L3MBTL1 (0.48) ALDH1A1KDM4EMAPTKMT2ADYRK1A
SCHEMBL1017994 0.68 DAO (0.51) KDM4EMAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104379560-A Benzamide derivative CHUGAI PHARMACEUTICAL CO LTD 2015-02-25 CN disclosed
CN-104379568-A Quinazolinedione derivative CHUGAI PHARMACEUTICAL CO LTD 2015-02-25 CN disclosed