SCHEMBL27997012

SCHEMBL27997012

CC(O)CC(C#N)c1cccc(C(F)(F)F)c1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PNMT P11086 1/20 0.50
CES2 O00748 1/20 0.43
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
HTR2B P41595 1/20 0.41
ACP3 P15309 2/20 0.40
CTSL P07711 1/20 0.40
EPHX1 P07099 2/20 0.39
DAO P14920 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
IDO1 P14902 1/20 0.38
TDO2 P48775 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
ATM Q13315 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL958288 0.82 PNMT (0.47) PNMTCES2HTR2AHTR2CHTR2B
SCHEMBL20521478 0.82 ACP3 (0.46) PNMTCES2ACP3CTSLEPHX1
SCHEMBL27997011 0.80 GPR139 (0.42) SLC6A2
SCHEMBL28816371 0.79 CYP11B1 (0.35) PNMTL3MBTL1
SCHEMBL28816314 0.79 CES2 (0.46) PNMTCES2ACP3CTSLEPHX1
SCHEMBL3913019 0.77 PNMT (0.47) PNMTCES2HTR2AHTR2CHTR2B
SCHEMBL11865382 0.76 TSHR (0.50) HTR2A
SCHEMBL343403 0.74 PNMT (0.61) PNMTCES2HTR2AHTR2CHTR2B
SCHEMBL1044909 0.74 PNMT (0.61) PNMTCES2HTR2AHTR2CHTR2B
SCHEMBL1535283 0.74 PNMT (0.61) PNMTCES2HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104254522-A Methanol derivatives as trpv3 modulators ABBVIE INC 2014-12-31 CN disclosed