SCHEMBL27997352

SCHEMBL27997352

CCOC(=O)COc1[c]ccc(Br)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C19 P33261 1/20 0.46
GAA P10253 2/20 0.42
NPSR1 Q6W5P4 1/20 0.42
KDM4E B2RXH2 3/20 0.41
HSD17B10 Q99714 1/20 0.41
POLB P06746 3/20 0.41
PABPC1 P11940 1/20 0.41
APOBEC3A P31941 1/20 0.41
APOBEC3G Q9HC16 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.39
PPARG P37231 1/20 0.39
PPARA Q07869 1/20 0.39
CASP3 P42574 1/20 0.39
CASP7 P55210 1/20 0.39
CASP9 P55211 1/20 0.39
TSHR P16473 2/20 0.38
USP2 O75604 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27997553 0.82 GAA (0.44) ALDH1A1CYP1A2GAANPSR1KDM4E
SCHEMBL7774207 0.79 HPGD (0.37) ALDH1A1GAAHSD17B10SMN1; SMN2TSHR
SCHEMBL1444265 0.77 ALDH1A1 (0.48) ALDH1A1GAANPSR1KDM4EHSD17B10
SCHEMBL16559854 0.74 ALDH1A1 (0.55) ALDH1A1CYP1A2CYP2C19GAAKDM4E
SCHEMBL1387968 0.74 GAA (0.42) ALDH1A1CYP1A2CYP2C19GAANPSR1
SCHEMBL7028752 0.73 ALDH1A1 (0.58) ALDH1A1CYP1A2CYP2C19GAANPSR1
SCHEMBL7033340 0.73 PPARA (0.59) ALDH1A1CYP2C19GAANPSR1KDM4E
SCHEMBL4517104 0.73 MEN1 (0.57) ALDH1A1NPSR1KDM4EPOLBPABPC1
SCHEMBL20564353 0.73 HPGD (0.41) ALDH1A1GAAKDM4EPOLBSMN1; SMN2
SCHEMBL12611682 0.72 GAA (0.55) ALDH1A1CYP1A2CYP2C19GAANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102958914-B 1-phenyl substituted heterocyclic derivatives and their use as prostaglandin D2 receptor modulators ACTELION PHARMACEUTICALS LTD 2015-05-27 CN disclosed
CN-104428305-A 1-phenyl-substituted heterocyclyl derivatives and their use as prostaglandin d2 receptor modulators ACTELION PHARMACEUTICALS LTD 2015-03-18 CN disclosed