SCHEMBL27997635

SCHEMBL27997635

[CH2]Cc1ccc(C)c(C)n1

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.44
NOS1 P29475 1/20 0.44
NOS2 P35228 1/20 0.44
ADORA2A P29274 1/20 0.30
ADORA1 P30542 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10730430 0.78 NOS3 (0.46) NOS3NOS1NOS2ADORA2AADORA1
SCHEMBL5517171 0.76 NOS3 (0.44) NOS3NOS1NOS2ADORA2AADORA1
SCHEMBL27778961 0.76 NOS3 (0.44) NOS3NOS1NOS2ADORA2AADORA1
SCHEMBL1161623 0.76 CCR1 (0.50) NOS3NOS1NOS2ADORA2AADORA1
SCHEMBL2125060 0.76 NOS3 (0.50) NOS3NOS1NOS2ADORA2AADORA1
SCHEMBL1161423 0.76 CCR1 (0.50) NOS3NOS1NOS2ADORA2AADORA1
Hydrochloric Acid SCHEMBL27554469 0.74 NOS3 (0.43) NOS3NOS1NOS2
SCHEMBL13809555 0.74 NOS2 (0.43) NOS3NOS1NOS2
SCHEMBL10647517 0.73 NOS3 (0.41) NOS3NOS1NOS2
SCHEMBL19413635 0.73 NOS3 (0.41) NOS3NOS1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102791714-B N-(imidazopyrimidin-7-yl)-heteroarylamide derivatives and their use as PDE10A inhibitors HOFFMANN LA ROCHE 2015-03-25 CN disclosed