SCHEMBL28002192

SCHEMBL28002192

CN(C)C1CCN(Cc2cc[c]c(F)c2)CC1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 4/20 0.46
MAP4K4 O95819 3/20 0.43
CCR3 P51677 1/20 0.41
TNKS O95271 1/20 0.39
PARP2 Q9UGN5 1/20 0.38
KCNH2 Q12809 3/20 0.38
CYP2D6 P10635 1/20 0.38
HRH1 P35367 1/20 0.38
GRM2 Q14416 1/20 0.37
EHMT2 Q96KQ7 1/20 0.37
ACHE P22303 1/20 0.37
GPR119 Q8TDV5 1/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28001856 0.92 MAP4K4 (0.45) PARP1MAP4K4CCR3HRH1GRM2
SCHEMBL1662326 0.79 ALDH1A1 (0.50) ALDH1A1
SCHEMBL23166113 0.75 HRH3 (0.50) PARP1ALDH1A1
SCHEMBL19311829 0.74 PARP1 (0.50) PARP1MAP4K4CCR3TNKSPARP2
SCHEMBL1661473 0.73 ALDH1A1 (0.33) GRM2ALDH1A1
SCHEMBL28444707 0.72 LMNA (0.52) KCNH2GRM2ALDH1A1
SCHEMBL2108897 0.72 ACHE (0.66) CCR3KCNH2ACHE
SCHEMBL1661217 0.72 S1PR5 (0.53) CCR3ALDH1A1
SCHEMBL1661451 0.72 S1PR5 (0.53) CCR3ALDH1A1
SCHEMBL1661132 0.72 S1PR5 (0.53) CCR3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104507933-B Amido quinazoline and Pyridopyrimidine derivatives 霍夫曼-拉罗奇有限公司 2017-10-31 CN claimed
CN-104507933-A Aminoquinazoline and pyridopyrimidine derivatives HOFFMANN LA ROCHE 2015-04-08 CN claimed