SCHEMBL28003149

SCHEMBL28003149

NC(=O)c1nccnc1-c1nccs1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 1/20 0.40
ECE1 P42892 1/20 0.39
ADORA2A P29274 6/20 0.39
LRRK2 Q5S007 1/20 0.39
ADORA1 P30542 6/20 0.38
ALDH1A1 P00352 2/20 0.36
PDPK1 O15530 1/20 0.36
LOXL2 Q9Y4K0 1/20 0.36
TGFBR1 P36897 1/20 0.36
HSP90AA1 P07900 1/20 0.35
TSHR P16473 1/20 0.34
NOS1 P29475 1/20 0.34
HSD17B10 Q99714 1/20 0.34
HDAC3 O15379 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC10 Q969S8 1/20 0.34
HDAC11 Q96DB2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29983575 0.75 PARP1 (0.46) CHEK2ECE1ADORA2AADORA1ALDH1A1
SCHEMBL2887102 0.75 CHEK2 (0.43) CHEK2ADORA2ALRRK2ADORA1PDPK1
SCHEMBL5597444 0.75 PARP1 (0.46) CHEK2ECE1ADORA2AADORA1ALDH1A1
SCHEMBL31238995 0.72 ERCC1 (0.47) CHEK2ALDH1A1TSHRHSD17B10
SCHEMBL3838752 0.71 ADORA2A (0.53) CHEK2ADORA2AADORA1ALDH1A1PDPK1
SCHEMBL2492969 0.71 TSHR (0.48) ADORA2AADORA1ALDH1A1PDPK1TSHR
SCHEMBL18113788 0.69 CHEK2 (0.50) CHEK2ECE1ADORA2AALDH1A1PDPK1
SCHEMBL6316389 0.69 CHEK2 (0.39) CHEK2ECE1ADORA2AADORA1ALDH1A1
SCHEMBL6649184 0.69 ADORA2A (0.41) CHEK2ECE1ADORA2ALRRK2ADORA1
SCHEMBL29290790 0.68 ECE1 (0.46) CHEK2ECE1ADORA2AADORA1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104254534-B Modulators of HEC1 activity and methods thereof 泰纬生命科技股份有限公司 2017-07-14 CN disclosed
CN-104395752-A Biomarkers for cancer responsive to modulators of HEC1 activity TAIVEX THERAPEUTICS CORP 2015-03-04 CN disclosed