SCHEMBL28004262

SCHEMBL28004262

NCc1ccc([C@@H]2CCNC2)cc1

nearest known ligand 0.59

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 1/20 0.59
JAK3 P52333 2/20 0.45
SLC18A3 Q16572 1/20 0.42
SIGMAR1 Q99720 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28003831 1.00 HTR3A (0.59) HTR3AJAK3SLC18A3SIGMAR1
SCHEMBL27815081 0.91 HTR3A (0.49) HTR3A
SCHEMBL27489026 0.89 SLC18A3 (0.55) HTR3ASLC18A3SIGMAR1
SCHEMBL28672856 0.86 HTR3A (0.56) HTR3AJAK3
SCHEMBL27511207 0.83 DRD2 (0.48) HTR3ASLC18A3SIGMAR1
SCHEMBL23763865 0.81 HTR3A (0.59) HTR3AJAK3
SCHEMBL27469424 0.81 HTR3A (0.59) HTR3AJAK3
SCHEMBL28258195 0.81 HTR3A (0.59) HTR3AJAK3
SCHEMBL17825381 0.79 HTR3A (0.56) HTR3AJAK3
SCHEMBL5839498 0.79 HTR3A (0.66) HTR3AJAK3SLC18A3SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104470918-A Aromatic heterocyclic derivative and pharmaceutical NIPPON SHINYAKU CO LTD 2015-03-25 CN disclosed