SCHEMBL28004656

SCHEMBL28004656

CS(=O)(=O)c1ccc(-c2cccnc2)nc1

nearest known ligand 0.60

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.60
CYP2A6 P11509 3/20 0.60
CYP3A4 P08684 1/20 0.60
PTGS1 P23219 4/20 0.53
CA12 O43570 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA9 Q16790 1/20 0.50
LMNA P02545 1/20 0.48
POLB P06746 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28146268 0.89 PTGS2 (0.64) PTGS2CYP2A6CYP3A4PTGS1CA12
SCHEMBL13589551 0.84 RORC (0.53) PTGS2PTGS1
SCHEMBL30846393 0.83 CA9 (0.68) PTGS2CYP2A6CYP3A4CA12CA1
SCHEMBL14378767 0.83 PTGS2 (0.48) PTGS2CYP3A4PTGS1CA12CA1
SCHEMBL18876343 0.81 PTGS2 (0.76) PTGS2CYP2A6CYP3A4PTGS1CA12
SCHEMBL12077434 0.78 GAA (0.55) CYP2A6CYP3A4CA12CA1CA2
SCHEMBL29497666 0.78 NAPRT (0.63) PTGS2CYP2A6CYP3A4PTGS1CA12
SCHEMBL355006 0.78 NAPRT (0.63) PTGS2CYP2A6CYP3A4PTGS1CA12
SCHEMBL8935802 0.76 CYP2A6 (0.69) CYP2A6CYP3A4CA12CA1CA2
Hydrochloric Acid SCHEMBL27577370 0.76 NAPRT (0.61) PTGS2PTGS1CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102639500-B Tricyclic compound, preparation method and pharmaceutical use thereof SHANGHAI HENGRUI PHARM CO LTD 2015-02-11 CN disclosed