SCHEMBL28004663

SCHEMBL28004663

CCn1cc(C=O)c(=O)c2ccc(N3CCNCC3)cc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
LMNA P02545 2/20 0.43
HTT P42858 2/20 0.43
KDM4E B2RXH2 1/20 0.43
BRD4 O60885 1/20 0.43
HPGD P15428 1/20 0.43
TSHR P16473 1/20 0.43
CYP2J2 P51589 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
HSD17B10 Q99714 1/20 0.43
KHK P50053 7/20 0.42
ADRB1 P08588 5/20 0.39
HTR6 P50406 3/20 0.39
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.37
CYP2C9 P11712 2/20 0.36
ATP6V1B2 P21281 1/20 0.36
TBXA2R P21731 1/20 0.36
EDNRA P25101 1/20 0.36
TARBP2 Q15633 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28005044 0.87 ALDH1A1 (0.43) ALDH1A1KDM4EBRD4HPGDKHK
SCHEMBL11711995 0.81 KDM4E (0.67) ALDH1A1LMNAHTTKDM4EBRD4
SCHEMBL13576340 0.80 KDM4E (0.69) ALDH1A1LMNAHTTKDM4EBRD4
SCHEMBL29724104 0.80 KDM4E (0.69) ALDH1A1LMNAHTTKDM4EBRD4
SCHEMBL11713505 0.77 LMNA (0.54) ALDH1A1LMNAHTTKDM4EBRD4
SCHEMBL22795618 0.72 ALDH1A1 (0.47) ALDH1A1HTTKDM4EBRD4KHK
SCHEMBL3973297 0.71 KDM4E (0.67) ALDH1A1LMNAHTTKDM4EBRD4
SCHEMBL21591573 0.71 MEN1 (0.57) ALDH1A1LMNAHTTHPGDMAPT
SCHEMBL14116369 0.70 CASP1 (0.54) ALDH1A1LMNAKDM4EHPGDTSHR
SCHEMBL6779177 0.69 KMT2A (0.60) ALDH1A1LMNAHTTKDM4EBRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104447537-B A kind of 3,3 '-methylene containing ethyl quinolinium ring-bis-fluoro quinolone derivatives and its preparation method and application 河南大学 2016-08-24 CN disclosed
CN-104447537-A 3,3'-methylene-bisfluoroquinolone derivative containing ethylquinoline rings as well as preparation method and application thereof UNIV HENAN 2015-03-25 CN disclosed