SCHEMBL28005447

SCHEMBL28005447

Cc1nc(CCBr)nc2ccccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
CYP1A2 P05177 3/20 0.50
HPGD P15428 2/20 0.50
GPR3 P46089 1/20 0.50
NUDT1 P36639 1/20 0.50
HSD17B10 Q99714 1/20 0.50
MPO P05164 1/20 0.42
RAD52 P43351 1/20 0.42
KDM4E B2RXH2 3/20 0.42
GAA P10253 1/20 0.42
POLB P06746 1/20 0.40
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
NPC1 O15118 2/20 0.38
MAPK1 P28482 2/20 0.38
TP53 P04637 1/20 0.38
MAPT P10636 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17194216 0.85 GPR3 (0.53) ALDH1A1CYP1A2HPGDGPR3NUDT1
SCHEMBL17904025 0.84 ALDH1A1 (0.56) ALDH1A1CYP1A2HPGDGPR3NUDT1
SCHEMBL14842813 0.81 ALDH1A1 (0.49) ALDH1A1CYP1A2HPGDGPR3NUDT1
SCHEMBL14985883 0.79 GPR3 (0.55) ALDH1A1CYP1A2HPGDGPR3NUDT1
SCHEMBL27871640 0.78 TLR8 (0.52) ALDH1A1CYP1A2HPGDGPR3NUDT1
SCHEMBL27871518 0.78 TLR8 (0.52) ALDH1A1CYP1A2HPGDGPR3NUDT1
SCHEMBL637147 0.78 GPR3 (0.53) ALDH1A1CYP1A2HPGDGPR3NUDT1
SCHEMBL16432784 0.78 GPR3 (0.53) ALDH1A1CYP1A2HPGDGPR3NUDT1
SCHEMBL29693664 0.78 GPR3 (0.53) ALDH1A1CYP1A2HPGDGPR3NUDT1
SCHEMBL19988074 0.78 GPR3 (0.53) ALDH1A1CYP1A2HPGDGPR3NUDT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105367572-B A kind of intermediate for preparing the compound as 4 inhibitor of dipeptidyl peptidase 浙江永太科技股份有限公司 2017-03-29 CN disclosed
CN-105503873-B Preparation method of chemical compound serving as DPP-IV (dipeptidyl peptidase-4) inhibitor 浙江永太科技股份有限公司 2017-03-22 CN disclosed
CN-104478880-B As the Biguanide derivative of DPP-IV inhibitor ZHEJIANG YONGTAI TECHNOLOGY CO., LTD. (CN) 2016-03-02 CN disclosed
CN-104478880-A Biguanide derivative as DPP-IV (dipeptidyl peptidase-4) inhibitor ZHEJIANG YONGTAI TECHNOLOGY CO LTD 2015-04-01 CN disclosed