SCHEMBL28005506

SCHEMBL28005506

CCc1ccc(-c2nc(N)sc2-c2cc(OC)c(OC)c(OC)c2)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.53
ADORA1 P30542 1/20 0.48
MAPT P10636 3/20 0.47
KDM4E B2RXH2 2/20 0.47
LMNA P02545 2/20 0.47
MAPK1 P28482 2/20 0.47
XBP1 P17861 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
TUBB1 Q9H4B7 3/20 0.44
PTGS2 P35354 1/20 0.43
ALDH1A1 P00352 3/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2D6 P10635 2/20 0.42
CYP2C19 P33261 2/20 0.42
TUBB4A P04350 2/20 0.42
TUBB P07437 2/20 0.42
TUBA3C P0DPH7 2/20 0.42
TUBA1B P68363 2/20 0.42
TUBA4A P68366 2/20 0.42
TUBB4B P68371 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28005543 0.90 ADORA1 (0.48) SMN1; SMN2ADORA1MAPTKDM4ELMNA
SCHEMBL28005196 0.85 TUBB4A (0.49) SMN1; SMN2ADORA1MAPTKDM4ELMNA
SCHEMBL28005179 0.84 ALDH1A1 (0.62) SMN1; SMN2ADORA1MAPTKDM4ELMNA
SCHEMBL28005220 0.84 TUBB4A (0.52) SMN1; SMN2ADORA1MAPTKDM4ELMNA
SCHEMBL28005576 0.80 KDM4E (0.50) SMN1; SMN2ADORA1MAPTKDM4ELMNA
SCHEMBL28005177 0.80 PDGFRB (0.50) SMN1; SMN2ADORA1MAPTKDM4ELMNA
SCHEMBL10120223 0.78 KDM4E (0.56) SMN1; SMN2ADORA1MAPTKDM4ELMNA
SCHEMBL28005174 0.77 ADORA1 (0.50) SMN1; SMN2ADORA1MAPTKDM4ELMNA
SCHEMBL5045105 0.76 SMN1; SMN2 (0.61) SMN1; SMN2MAPTKDM4ELMNAMAPK1
SCHEMBL10120710 0.75 KDM4E (0.53) SMN1; SMN2ADORA1MAPTKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104418821-A 2, 4-substituted 5- (3,4, 5-trimethoxyphenyl) thiazole derivative and preparation method and application thereof WEST CHINA HOSPITAL SICHUAN UNIV 2015-03-18 CN claimed
CN-104418821-A 2, 4-substituted 5- (3,4, 5-trimethoxyphenyl) thiazole derivative and preparation method and application thereof WEST CHINA HOSPITAL SICHUAN UNIV 2015-03-18 CN disclosed