SCHEMBL28006307

SCHEMBL28006307

C=CC(=O)OCCCNC(=O)CNC(=O)OC(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA1 P00915 8/20 0.46
CA2 P00918 8/20 0.46
CA12 O43570 7/20 0.46
CA9 Q16790 7/20 0.46
TSHR P16473 5/20 0.44
HPGD P15428 1/20 0.44
ALDH1A1 P00352 3/20 0.44
CYP3A4 P08684 1/20 0.44
TDP1 Q9NUW8 1/20 0.43
MAOA P21397 1/20 0.42
MAOB P27338 1/20 0.42
MEN1 O00255 1/20 0.41
GAA P10253 1/20 0.41
KMT2A Q03164 1/20 0.41
THRB P10828 1/20 0.38
TP53 P04637 2/20 0.37
HIF1A Q16665 2/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL759464 0.90 CA12 (0.55) CA1CA2CA12CA9TSHR
SCHEMBL759467 0.86 CA12 (0.61) CA1CA2CA12CA9TSHR
SCHEMBL4138078 0.85 CA12 (0.62) CA1CA2CA12CA9TSHR
SCHEMBL757089 0.81 TDP1 (0.47) CA1CA2CA12CA9TSHR
SCHEMBL14723706 0.79 TDP1 (0.66) CA1CA2CA12CA9ALDH1A1
SCHEMBL18510208 0.79 MAOA (0.50) CA1CA2CA12CA9TSHR
SCHEMBL18352554 0.78 CA12 (0.57) CA1CA2CA12CA9TDP1
SCHEMBL16450357 0.77 CA12 (0.54) CA1CA2CA12CA9TDP1
SCHEMBL17884326 0.77 TDP1 (0.42) CA1CA2CA12CA9TSHR
SCHEMBL8156813 0.76 TSHR (0.59) TSHRHPGDALDH1A1CYP3A4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102460221-B Biomedical devices BAUSCH & LOMB 2015-04-01 CN disclosed