SCHEMBL28008334

SCHEMBL28008334

Cc1cc(F)c(F)cc1Cn1cc(C(N)=O)cn1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 12/20 0.44
L3MBTL1 Q9Y468 2/20 0.43
ALDH1A1 P00352 2/20 0.43
MAPT P10636 1/20 0.43
PKM P14618 1/20 0.43
ACHE P22303 2/20 0.39
GRM2 Q14416 3/20 0.38
NR1I2 O75469 1/20 0.37
KCNH2 Q12809 1/20 0.37
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25381150 0.87 L3MBTL1 (0.42) KLKB1L3MBTL1ALDH1A1MAPTPKM
SCHEMBL28818252 0.79 KLKB1 (0.49) KLKB1L3MBTL1ALDH1A1MAPTPOLB
SCHEMBL28008768 0.79 MAPT (0.48) KLKB1L3MBTL1ALDH1A1MAPTPOLB
SCHEMBL28008774 0.79 KLKB1 (0.47) KLKB1GRM2NR1I2KCNH2
SCHEMBL28818254 0.78 KLKB1 (0.53) KLKB1ALDH1A1MAPTGRM2
SCHEMBL20481563 0.78 ALDH1A1 (0.51) KLKB1L3MBTL1ALDH1A1MAPTPKM
SCHEMBL28008833 0.77 KLKB1 (0.46) KLKB1L3MBTL1
SCHEMBL1416055 0.77 KLKB1 (0.55) KLKB1L3MBTL1ALDH1A1MAPTGRM2
SCHEMBL27364065 0.76 KLKB1 (0.41) KLKB1L3MBTL1ALDH1A1MAPTPKM
SCHEMBL28008344 0.76 KLKB1 (0.48) KLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103080104-B N-((6-amino-pyridin-3-yl)methyl)-heteroaryl-carboxamides as inhibitors of plasma kallikrein NOVARTIS AG 2015-04-08 CN claimed
CN-103080104-B N-((6-amino-pyridin-3-yl)methyl)-heteroaryl-carboxamides as inhibitors of plasma kallikrein NOVARTIS AG 2015-04-08 CN disclosed