SCHEMBL2801676

SCHEMBL2801676

CC(C)(C)OC(=O)NS(=O)(=O)N1CCC(=O)CC1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.39
CA14 Q9ULX7 4/20 0.39
CA1 P00915 2/20 0.39
CA7 P43166 2/20 0.39
CA2 P00918 1/20 0.39
CCNT1 O60563 1/20 0.37
CDK9 P50750 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
NFKB1 P19838 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
STS P08842 1/20 0.33
GAA P10253 1/20 0.33
BRS3 P32247 1/20 0.32
CTSK P43235 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12792779 0.83 CA12 (0.42) CA12CA14CA1CA7CA2
SCHEMBL583414 0.83 CA12 (0.42) CA12CA14CA1CA7CA2
SCHEMBL12421750 0.82 CA12 (0.45) CA12CA14CA1CA7CA2
SCHEMBL3936868 0.81 CA12 (0.41) CA12CA14CA1CA7CA2
SCHEMBL17057869 0.79 CA12 (0.40) CA12CA14CA1CA7CA2
SCHEMBL4177994 0.79 SMN1; SMN2 (0.47) CA12CA14CA1CA7CA2
SCHEMBL13610628 0.78 STS (0.47) STS
SCHEMBL22404282 0.78 CA12 (0.39) CA12CA14CA1CA7CA2
SCHEMBL21775398 0.77 KDM1A (0.37)
SCHEMBL1819405 0.77 CA12 (0.40) CA12CA14CA1CA7CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3095784-A1 APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES AbbVie Inc. (US) 2016-11-23 EP disclosed
US-9493431-B2 Apoptosis-inducing agent for the treatment of cancer and immune and autoimmune diseases ABBVIE INC. (US) 2016-11-15 US disclosed
EP-2387559-B1 APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES ABBVIE INC (US) 2016-06-29 EP disclosed
US-20160002187-A1 APOPTOSIS-INDUCING AGENT FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES ABBVIE INC (US) 2016-01-07 US disclosed
US-9156856-B2 Apoptosis-inducing agents for the treatment of cancer and immune and autoimmune diseases ABBVIE INC. (US) 2015-10-13 US disclosed
US-20130184278-A1 APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES ABBOTT LABORATORIES (US) 2013-07-18 US disclosed
US-8338466-B2 Apoptosis-inducing agents for the treatment of cancer and immune and autoimmune diseases ABBOTT LABORATORIES (US) 2012-12-25 US disclosed
US-7772225-B2 N-sulfamoyl-piperidineamides for the treatment or inhibition of obesity and related conditions SOLVAY PHARMACEUTICALS GMBH (DE) 2010-08-10 US disclosed
US-7772225-B2 N-sulfamoyl-piperidineamides for the treatment or inhibition of obesity and related conditions SOLVAY PHARMACEUTICALS GMBH (DE) 2010-08-10 US disclosed
US-20100184766-A1 APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES ABBOTT LABORATORIES (US) 2010-07-22 US disclosed
US-20070149512-A1 N-Sulfamoyl-piperidineamides for the treatment or inhibition of obesity and related conditions SOLVAY PHARMACEUTICALS GMBH 2007-06-28 US disclosed
US-20070149512-A1 N-Sulfamoyl-piperidineamides for the treatment or inhibition of obesity and related conditions SOLVAY PHARMACEUTICALS GMBH 2007-06-28 US disclosed
WO-2007065948-A1 NOVEL N-SULFAMOYL-PIPERIDINEAMIDES FOR THE PROPHYLAXIS OR TREATMENT OF OBESITY AND RELATED CONDITIONS SOLVAY PHARMACEUTICALS GMBH (DE) 2007-06-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070149512-A1 N-Sulfamoyl-piperidineamides for the treatment or inhibition of obesity and related conditions FABP4, GPR119, SRM CA12 4141/4885CA14 4318/4885CA1 4320/4885
US-20100184766-A1 APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES BCL2, BAX, BCL3 CA12 1100/4885CA14 1303/4885CA1 1290/4885
US-20160002187-A1 APOPTOSIS-INDUCING AGENT FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES BCL2, BAX, BCL3 CA12 1019/4885CA14 1288/4885CA1 1330/4885
US-20130184278-A1 APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES BCL2, BAX, BCL3 CA12 1100/4885CA14 1303/4885CA1 1290/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.