SCHEMBL28017809

SCHEMBL28017809

Cc1cc(C)cc(OC(C)CC#N)c1

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.39
ALDH1A1 P00352 2/20 0.32
CYP3A4 P08684 1/20 0.32
TSHR P16473 1/20 0.32
MAPK1 P28482 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28263637 0.74 MTNR1A (0.46)
SCHEMBL9774796 0.74 TP53 (0.36) ALDH1A1CYP3A4TSHRMAPK1TDP1
SCHEMBL2107806 0.72 ALDH1A1 (0.42) ALDH1A1SMN1; SMN2
SCHEMBL2107809 0.72 ALDH1A1 (0.42) ALDH1A1SMN1; SMN2
SCHEMBL14465627 0.71 GPBAR1 (0.38) ALDH1A1CYP3A4TSHRMAPK1TDP1
SCHEMBL25059065 0.71 MTNR1A (0.35) ALDH1A1CYP3A4TSHRMAPK1TDP1
SCHEMBL21207860 0.71 MTNR1A (0.35) ALDH1A1CYP3A4TSHRMAPK1TDP1
SCHEMBL5291180 0.69 ALDH1A1 (0.42) ALDH1A1CYP3A4TSHRMAPK1TDP1
SCHEMBL12285479 0.69 ALDH1A1 (0.42) ALDH1A1CYP3A4TSHRMAPK1TDP1
SCHEMBL12329328 0.69 OPRM1 (0.33) ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104684907-A Antidiabetic tricyclic compounds MERCK SHARP & DOHME 2015-06-03 CN disclosed