SCHEMBL28020076

SCHEMBL28020076

CC(=O)/C(C(=O)OC(C)C)=C(\NCc1ccccc1)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.48
CYP2D6 P10635 1/20 0.44
ALDH1A1 P00352 4/20 0.43
MAPT P10636 2/20 0.43
MEN1 O00255 2/20 0.43
TSHR P16473 1/20 0.43
HPGD P15428 3/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
MME P08473 1/20 0.42
TP53 P04637 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA3 P07451 1/20 0.41
CA4 P22748 1/20 0.41
CA6 P23280 1/20 0.41
CA5A P35218 1/20 0.41
CA7 P43166 1/20 0.41
CACNA1C Q13936 1/20 0.41
SCN9A Q15858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28020080 1.00 KMT2A (0.48) KMT2ACYP2D6ALDH1A1MAPTMEN1
SCHEMBL28820145 0.85 KMT2A (0.46) KMT2ACYP2D6ALDH1A1MAPTMEN1
SCHEMBL28820146 0.85 KMT2A (0.46) KMT2ACYP2D6ALDH1A1MAPTMEN1
SCHEMBL28020416 0.83 PPID (0.50) KMT2ACYP2D6ALDH1A1MAPTMEN1
SCHEMBL28020411 0.83 PPID (0.50) KMT2ACYP2D6ALDH1A1MAPTMEN1
SCHEMBL28019981 0.82 CYP2C9 (0.50) KMT2ACYP2D6ALDH1A1MAPTMEN1
SCHEMBL28019983 0.82 CYP2C9 (0.50) KMT2ACYP2D6ALDH1A1MAPTMEN1
SCHEMBL28020429 0.82 LMNA (0.45) KMT2AALDH1A1HPGDTP53CA12
SCHEMBL28020432 0.82 LMNA (0.45) KMT2AALDH1A1HPGDTP53CA12
SCHEMBL19500095 0.77 KMT2A (0.61) KMT2AALDH1A1MAPTMEN1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103910644-B Beta-enaminone ester compounds, and synthesis method and application of beta-enaminone ester compounds UNIV GUANGXI NORMAL 2015-06-24 CN disclosed