SCHEMBL28020890

SCHEMBL28020890

CCS(=O)(=O)c1ccc(C(F)F)cc1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PSIP1 O75475 2/20 0.52
GAA P10253 1/20 0.52
RORC P51449 10/20 0.42
RORA P35398 3/20 0.40
ALDH1A1 P00352 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
PTGS2 P35354 1/20 0.36
KIF11 P52732 1/20 0.36
TRPV4 Q9HBA0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10455034 0.81 PSIP1 (0.74) PSIP1GAAALDH1A1CYP3A4CYP2C9
SCHEMBL10180779 0.80 GAA (0.59) PSIP1GAARORCALDH1A1
SCHEMBL16441817 0.78 PSIP1 (0.52) PSIP1GAARORCRORAALDH1A1
SCHEMBL19987486 0.78 PSIP1 (0.52) PSIP1GAARORCRORAALDH1A1
SCHEMBL17289163 0.77 ENPP2 (0.50) CYP3A4PTGS2
SCHEMBL30026174 0.77 PSIP1 (0.50) PSIP1GAARORCRORAALDH1A1
SCHEMBL18440551 0.77 GAA (0.55) PSIP1GAARORCRORAALDH1A1
SCHEMBL28554996 0.77 PSIP1 (0.50) PSIP1GAARORCRORAALDH1A1
SCHEMBL10179790 0.77 PSIP1 (0.50) PSIP1GAAALDH1A1
SCHEMBL16232116 0.77 GAA (0.55) PSIP1GAARORCRORAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104837843-A Imidazopyridazine derivatives as GABAA receptor modulators PFIZER 2015-08-12 CN disclosed