SCHEMBL28020910

SCHEMBL28020910

COc1cc(CN2C(=O)CCC2C(N)=O)cc(OC)c1

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 7/20 0.45
HCRTR2 O43614 7/20 0.45
KMT2A Q03164 6/20 0.43
GYS1 P13807 1/20 0.42
TDP1 Q9NUW8 1/20 0.41
SIGMAR1 Q99720 1/20 0.40
MEN1 O00255 1/20 0.40
KDM4E B2RXH2 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL289561 0.90 GYS1 (0.49) HCRTR1HCRTR2KMT2AGYS1TDP1
SCHEMBL289122 0.90 GYS1 (0.49) HCRTR1HCRTR2KMT2AGYS1TDP1
SCHEMBL28020905 0.87 HCRTR1 (0.53) HCRTR1HCRTR2KMT2AGYS1KDM4E
SCHEMBL28020907 0.81 P2RX7 (0.45) HCRTR2KMT2AGYS1MEN1
SCHEMBL288451 0.78 GYS1 (0.58) HCRTR1HCRTR2KMT2AGYS1SIGMAR1
SCHEMBL1612182 0.78 GYS1 (0.58) HCRTR1HCRTR2KMT2AGYS1SIGMAR1
SCHEMBL1162612 0.77 P2RX7 (0.54) KMT2A
SCHEMBL1162700 0.77 P2RX7 (0.54) KMT2A
SCHEMBL28270409 0.77 P2RX7 (0.54) KMT2A
SCHEMBL16600994 0.77 KMT2A (0.55) HCRTR1HCRTR2KMT2AGYS1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102482212-B Carboxamide compounds and they are as the purposes of calpain inhibitor ABBVIE (US) 2015-08-26 CN claimed
CN-102482212-B Carboxamide compounds and they are as the purposes of calpain inhibitor ABBVIE (US) 2015-08-26 CN disclosed