SCHEMBL28021031

SCHEMBL28021031

N#Cc1cccc(CN2C(=O)C=C[C@@H]2C(=O)O)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 1/20 0.46
FEN1 P39748 1/20 0.44
FAAH O00519 1/20 0.43
ALDH1A1 P00352 1/20 0.43
ADRA1D P25100 1/20 0.42
SIRT2 Q8IXJ6 1/20 0.42
SIRT1 Q96EB6 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
CYP19A1 P11511 1/20 0.40
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
VNN1 O95497 1/20 0.40
LMNA P02545 1/20 0.40
CREBBP Q92793 1/20 0.39
IDH1 O75874 1/20 0.39
FFAR1 O14842 1/20 0.39
FFAR4 Q5NUL3 1/20 0.39
FOLH1 Q04609 1/20 0.39
CCR3 P51677 1/20 0.39
MEP1A Q16819 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1613572 0.74 GYS1 (0.50) CCR2FEN1FAAHSIRT2SIRT1
SCHEMBL288654 0.74 GYS1 (0.50) CCR2FEN1FAAHSIRT2SIRT1
SCHEMBL7415511 0.73 SIRT2 (0.50) CCR2FEN1FAAHALDH1A1ADRA1D
SCHEMBL29586287 0.72 MGLL (0.55) CCR2FEN1FAAHALDH1A1ADRA1D
SCHEMBL28563919 0.72 MGLL (0.55) CCR2FEN1FAAHALDH1A1ADRA1D
SCHEMBL8443442 0.69 CCR2 (0.56) CCR2FEN1FAAHALDH1A1ADRA1D
SCHEMBL8872921 0.69 KMT2A (0.51) CCR2FAAH
SCHEMBL25395450 0.69 CCR2 (0.55) CCR2FEN1FAAHALDH1A1ADRA1D
SCHEMBL19401544 0.68 GYS1 (0.54) CCR2FAAHSIRT2SIRT1CCR3
SCHEMBL1764734 0.68 GYS1 (0.54) CCR2FAAHSIRT2SIRT1CCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102482212-B Carboxamide compounds and they are as the purposes of calpain inhibitor ABBVIE (US) 2015-08-26 CN disclosed