SCHEMBL28021758

SCHEMBL28021758

Cn1c(NC(=O)O)nc2cc(OCc3ccccc3)ccc21

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 2/20 0.58
SRD5A2 P31213 1/20 0.57
MEN1 O00255 5/20 0.55
KMT2A Q03164 5/20 0.55
NPC1 O15118 2/20 0.55
RAB9A P51151 2/20 0.55
BRAF P15056 3/20 0.51
ACSL1 P33121 1/20 0.48
HSP90AA1 P07900 1/20 0.47
PTGES O14684 1/20 0.46
RAF1 P04049 1/20 0.46
MAPT P10636 1/20 0.46
CYP3A4 P08684 1/20 0.46
BRD4 O60885 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5579673 0.79 PTGES (0.64) HDAC6SRD5A2MEN1KMT2ANPC1
SCHEMBL5349165 0.76 BRAF (0.49) BRAFRAF1
SCHEMBL8305123 0.75 HTR3A (0.54) SRD5A2MEN1KMT2ANPC1RAB9A
SCHEMBL3771751 0.74 RAB9A (0.74) HDAC6MEN1KMT2ANPC1RAB9A
SCHEMBL22382419 0.74 EHMT2 (0.53) HDAC6NPC1RAB9A
SCHEMBL19058673 0.74 HDAC6 (1.00) HDAC6
SCHEMBL4464733 0.73 SRD5A2 (0.81) SRD5A2MEN1KMT2ANPC1RAB9A
SCHEMBL4470968 0.73 SRD5A2 (1.00) SRD5A2MEN1KMT2ANPC1RAB9A
SCHEMBL6320502 0.72 HDAC6 (0.53) HDAC6NPC1RAB9AMAPT
SCHEMBL457343 0.72 TP53 (0.52) HDAC6MEN1KMT2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104876878-B - 2 alkyl substituted urea benzimidazoles compound of 5- aryl phenols and its application 中国科学院广州生物医药与健康研究院 2018-04-27 CN disclosed
CN-104876878-A 5-aryl phenol-2 alkyl substituted urea benzimidazole compound and applications thereof GUANGZHOU INST BIOMED & HEALTH 2015-09-02 CN disclosed