SCHEMBL28021938

SCHEMBL28021938

CNc1ccc(N2CCC(N(C)C)C2)c(C(F)(F)F)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EML4 Q9HC35 1/20 0.48
ALK Q9UM73 1/20 0.48
HSD11B1 P28845 2/20 0.43
CSF1R P07333 1/20 0.41
CDK4 P11802 1/20 0.41
CDK6 Q00534 1/20 0.41
TRPV1 Q8NER1 2/20 0.40
WDR5 P61964 2/20 0.40
FPR1 P21462 1/20 0.39
FPR2 P25090 1/20 0.39
CYP2C9 P11712 1/20 0.39
MCHR1 Q99705 2/20 0.38
SOS1 Q07889 2/20 0.38
HRH4 Q9H3N8 2/20 0.38
HRH3 Q9Y5N1 2/20 0.38
CCNA2 P20248 1/20 0.38
CDK2 P24941 1/20 0.38
CCNA1 P78396 1/20 0.38
LCK P06239 2/20 0.37
KDR P35968 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27959375 1.00 EML4 (0.48) EML4ALKHSD11B1CSF1RCDK4
SCHEMBL1749264 0.85 FPR1 (0.48) CSF1RCDK4CDK6WDR5FPR1
SCHEMBL1749267 0.85 FPR1 (0.48) CSF1RCDK4CDK6WDR5FPR1
SCHEMBL17135166 0.83 EML4 (0.47) EML4ALKHSD11B1TRPV1WDR5
SCHEMBL274575 0.83 EML4 (0.47) EML4ALKHSD11B1TRPV1WDR5
SCHEMBL3314851 0.78 EML4 (0.51) EML4ALKHSD11B1WDR5CYP2C9
SCHEMBL28027728 0.77 S1PR1 (0.50) CDK4CCNA2CDK2CCNA1PIM1
SCHEMBL1749702 0.76 MCHR1 (0.55) MCHR1HRH3
SCHEMBL282609 0.76 HRH4 (0.39) EML4ALKHSD11B1TRPV1WDR5
SCHEMBL13958468 0.75 TP53 (0.56) CSF1RCYP2C9CCNA2CDK2CCNA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104797581-A HETEROARYL ALKYNE COMPOUND AND APPLICATION THEREOF NANJING SANHOME PHARMACEUTICAL CO LTD 2015-07-22 CN disclosed