SCHEMBL28022336

SCHEMBL28022336

CC(C)(C)OC(=O)[C@H]1C(C(=O)O)CN2CCCC12

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 5/20 0.36
HSD17B10 Q99714 1/20 0.36
BTK Q06187 1/20 0.35
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
ALDH1A1 P00352 2/20 0.33
ADRA2A P08913 1/20 0.33
ADRA1A P35348 1/20 0.33
MAPT P10636 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
PDE4B Q07343 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27933965 0.80 ALDH1A1 (0.38) MEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL28022831 0.78 MEN1 (0.39) BTKMEN1KMT2AALDH1A1ADRA2A
SCHEMBL28022338 0.78 MEN1 (0.39) BTKMEN1KMT2AALDH1A1ADRA2A
SCHEMBL28288979 0.74 HRH3 (0.36) HSD17B10HRH3
SCHEMBL1297246 0.72 BTK (0.45) HSD17B10BTKMEN1KMT2AHRH3
SCHEMBL17336143 0.69 CHRM2 (0.48) GPR119HSD17B10MEN1KMT2AALDH1A1
SCHEMBL15369037 0.68 BTK (0.41) GPR119BTKALDH1A1HRH3
SCHEMBL23004339 0.68 BTK (0.47) HSD17B10BTKMEN1KMT2A
SCHEMBL1296980 0.68 BTK (0.44) BTKALDH1A1SMN1; SMN2
SCHEMBL15023147 0.68 BTK (0.47) HSD17B10BTKMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104703980-A Orexin receptor antagonists which are [ortho bi (hetero )aryl]-[2-(meta bi (hetero )aryl)-pyrrolidin-1-yl]-methanone derivatives ACTELION PHARMACEUTICALS LTD 2015-06-10 CN disclosed