SCHEMBL28022375

SCHEMBL28022375

COc1ccc(C(C)(C)CO)cc1S(N)(=O)=O

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.55
CA2 P00918 3/20 0.44
CA9 Q16790 3/20 0.44
CA12 O43570 2/20 0.44
CA1 P00915 2/20 0.44
TDP1 Q9NUW8 1/20 0.44
ALDH1A1 P00352 3/20 0.42
CA4 P22748 1/20 0.42
HTT P42858 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
GAA P10253 1/20 0.42
CNR1 P21554 1/20 0.41
CNR2 P34972 1/20 0.41
BRD4 O60885 1/20 0.40
WDR5 P61964 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8048512 0.88 PKM (0.51) PKMCA2CA9CA12CA1
SCHEMBL31525849 0.86 PKM (0.50) PKMCA2CA9CA12CA1
SCHEMBL21962105 0.85 PKM (0.59) PKMCA2CA9CA12CA1
SCHEMBL29469839 0.83 CA2 (0.57) PKMCA2CA9CA12CA1
SCHEMBL2446085 0.83 CA2 (0.57) PKMCA2CA9CA12CA1
SCHEMBL31172585 0.82 PKM (0.52) PKMCA2CA9CA12CA1
SCHEMBL35406099 0.81 PKM (0.54) PKMCA2CA9CA12CA1
SCHEMBL5189382 0.81 PKM (0.54) PKMCA2CA9CA12CA1
SCHEMBL31172598 0.79 PKM (0.44) PKMCA2CA9CA12CA1
SCHEMBL31525811 0.79 PKM (0.56) PKMCA2CA9CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105102449-B Antiviral compound 豪夫迈·罗氏有限公司 2017-06-13 CN disclosed
CN-105102449-A Antiviral compounds HOFFMANN LA ROCHE 2015-11-25 CN disclosed