SCHEMBL28022901

SCHEMBL28022901

CN(C(=O)c1cccc(-c2ccccc2)c1)C(F)(F)F

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 1/20 0.51
PDK2 Q15119 1/20 0.49
HDAC8 Q9BY41 1/20 0.47
ERN1 O75460 3/20 0.46
KEAP1 Q14145 1/20 0.44
NFE2L2 Q16236 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
ERCC5 P28715 1/20 0.44
FEN1 P39748 1/20 0.44
HSD17B2 P37059 3/20 0.44
HSD17B1 P14061 2/20 0.44
LMNA P02545 1/20 0.43
HPGD P15428 1/20 0.43
TSHR P16473 1/20 0.43
RXRA P19793 1/20 0.43
RXRB P28702 1/20 0.43
PRSS1 P07477 1/20 0.42
PRSS2 P07478 1/20 0.42
PRSS3 P35030 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20812226 0.85 KMO (0.53) KMOPDK2HDAC8ERN1MEN1
SCHEMBL6279720 0.84 NR1H3 (0.50) KMT2AHPGDTSHR
Trifluoroacetic Acid SCHEMBL5067780 0.83 PDK2 (0.57) KMOPDK2HDAC8ERN1KEAP1
SCHEMBL30283775 0.81 ERN1 (0.60) KMOPDK2HDAC8ERN1KEAP1
SCHEMBL1135975 0.81 ERN1 (0.60) KMOPDK2HDAC8ERN1KEAP1
Hydrochloric Acid SCHEMBL28646857 0.80 ERN1 (0.59) KMOPDK2HDAC8ERN1KEAP1
SCHEMBL28022357 0.78 KMO (0.56) KMOHDAC8ERN1MEN1KMT2A
Trimethylammonium SCHEMBL27623058 0.75 KMO (0.81) KMOHDAC8ERN1KEAP1ERCC5
SCHEMBL772236 0.75 KMO (0.53) KMOHDAC8ERN1MEN1KMT2A
SCHEMBL4434800 0.73 HPGD (0.73) KMOHDAC8ERCC5FEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105102449-A Antiviral compounds HOFFMANN LA ROCHE 2015-11-25 CN disclosed