SCHEMBL28024470

SCHEMBL28024470

c1cncc(-c2ccc3c(n2)CCCC3)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 4/20 0.55
CYP11B2 P19099 4/20 0.55
CYP2A6 P11509 4/20 0.46
HSP90AA1 P07900 1/20 0.45
HSP90AB1 P08238 1/20 0.45
PTK2 Q05397 1/20 0.45
CHRNB4 P30926 1/20 0.45
CHRNA3 P32297 1/20 0.45
CYP1A2 P05177 3/20 0.44
CYP3A4 P08684 3/20 0.44
ALDH1A1 P00352 2/20 0.44
CYP19A1 P11511 2/20 0.44
NPY5R Q15761 3/20 0.43
CYP2C19 P33261 2/20 0.42
THRB P10828 1/20 0.42
NPC1 O15118 1/20 0.42
CYP2C9 P11712 1/20 0.42
AXL P30530 1/20 0.41
PBRM1 Q86U86 1/20 0.41
MKNK1 Q9BUB5 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4195132 0.83 CHRNB2 (0.44) CYP11B1CYP11B2CYP2A6HSP90AA1HSP90AB1
SCHEMBL3310894 0.81 MEN1 (0.45) ALDH1A1NPC1MAPTKDM4ETSHR
SCHEMBL3247157 0.80 CYP2A6 (0.43) CYP11B1CYP11B2CYP2A6HSP90AA1HSP90AB1
SCHEMBL31598494 0.80 MEN1 (0.44) ALDH1A1NPC1MAPTKDM4ETSHR
SCHEMBL8283777 0.77 CYP1A2 (0.50) CYP11B1CYP11B2CYP2A6HSP90AA1HSP90AB1
SCHEMBL29648993 0.76 ADRA2A (0.50) ALDH1A1NPC1MAPTTSHRHSD17B10
SCHEMBL28540727 0.72 CYP2A6 (0.47) CYP11B1CYP11B2CYP2A6HSP90AA1HSP90AB1
SCHEMBL11641022 0.71 NPC1 (0.48) ALDH1A1NPC1MAPTKDM4EHTT
SCHEMBL3869454 0.71 KMT2A (0.41) CYP1A2ALDH1A1NPC1MAPTKDM4E
SCHEMBL10430601 0.71 ADRA2A (0.44) CYP3A4ALDH1A1NPC1MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104755471-A Pyridine derivative and drug NIPPON SHINYAKU CO LTD 2015-07-01 CN disclosed