SCHEMBL28024975

SCHEMBL28024975

Brc1ccc(CSc2ccc3ccccc3c2)cc1

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAOB P27338 6/20 0.57
MAOA P21397 3/20 0.53
CYP2A6 P11509 2/20 0.50
ANPEP P15144 1/20 0.46
CYP1A2 P05177 1/20 0.41
MGAM O43451 2/20 0.41
GAA P10253 2/20 0.41
SI P14410 2/20 0.41
MGAM2 Q2M2H8 2/20 0.41
KDM4E B2RXH2 1/20 0.41
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6057087 0.85 MAOA (0.58) MAOBMAOAANPEPRAB9A
SCHEMBL31468135 0.84 MAOB (0.50) MAOBMAOACYP2A6ANPEPRAB9A
SCHEMBL28024503 0.83 CYP2A6 (0.47) MAOBMAOACYP2A6ANPEP
SCHEMBL28386710 0.82 MAOB (0.57) MAOBMAOACYP2A6ANPEPCYP1A2
SCHEMBL28389508 0.82 MAOA (0.57) MAOBMAOACYP2A6ANPEPRAB9A
SCHEMBL20780451 0.82 CYP2A6 (0.50) MAOBMAOACYP2A6ANPEPCYP1A2
SCHEMBL28024991 0.80 MAOB (0.51) MAOBMAOAMGAMGAASI
SCHEMBL845713 0.79 MAOB (0.59) MAOBMAOACYP1A2
SCHEMBL19422820 0.78 MAOA (0.41) MAOBMAOACYP2A6ANPEPCYP1A2
SCHEMBL31307765 0.77 CYP1A2 (0.44) MAOBMAOACYP2A6ANPEPCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104892471-B Substance having protein tyrosine kinase inhibitory activity, preparation method and use thereof 中国人民解放军军事医学科学院放射与辐射医学研究所 2020-03-27 CN disclosed
CN-104892471-A Substances having protein tyrosine kinase inhibitory activity, and preparation method and use thereof INST RADIATION MED AMMS PLA 2015-09-09 CN disclosed