SCHEMBL28024503

SCHEMBL28024503

Brc1cccc(CSc2ccc3ccccc3c2)c1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.47
MAOB P27338 3/20 0.46
USP2 O75604 1/20 0.45
HPGD P15428 1/20 0.45
TSHR P16473 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
ANPEP P15144 1/20 0.44
PTGDR2 Q9Y5Y4 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
SIRT2 Q8IXJ6 1/20 0.41
MAOA P21397 1/20 0.41
CDC7 O00311 2/20 0.41
DBF4 Q9UBU7 2/20 0.41
HTT P42858 1/20 0.41
TAAR1 Q96RJ0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30418101 0.85 TAAR1 (0.47) CYP2A6MAOBANPEPMAOATAAR1
SCHEMBL28024975 0.83 MAOB (0.57) CYP2A6MAOBANPEPMAOA
SCHEMBL16143105 0.82 HTT (0.54) MAOBUSP2HPGDTSHRL3MBTL1
SCHEMBL6057087 0.82 MAOA (0.58) MAOBANPEPMAOA
SCHEMBL31468135 0.81 MAOB (0.50) CYP2A6MAOBANPEPMAOAHTT
SCHEMBL28024514 0.80 ALDH1A1 (0.51) CYP2A6HPGDL3MBTL1PTGDR2MEN1
SCHEMBL28386633 0.80 DAO (0.49) CYP2A6MAOBUSP2HPGDL3MBTL1
SCHEMBL28386632 0.80 RAB9A (0.53) CYP2A6MAOBHPGDL3MBTL1MEN1
SCHEMBL1710411 0.79 MAPT (0.54) MAOBMEN1KMT2AMAOAHTT
SCHEMBL19629067 0.79 MAOA (0.41) CYP2A6MAOBHPGDANPEPMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104892471-B Substance having protein tyrosine kinase inhibitory activity, preparation method and use thereof 中国人民解放军军事医学科学院放射与辐射医学研究所 2020-03-27 CN disclosed
CN-104892471-A Substances having protein tyrosine kinase inhibitory activity, and preparation method and use thereof INST RADIATION MED AMMS PLA 2015-09-09 CN disclosed